Ileal bile acid transporter inhibition, CYP7A1 induction, and antilipemic action of 264W94

Journal of Lipid Research

Volumn 43, Issue 8, 2002, Pages 1320-1330

  Root, Carolyn ^a   Smith, Chari D ^a   Sundseth, Scott S ^a   Pink, Heather M ^a   Wilson, Joan G ^a   Lewis, Michael C ^a  

^a GLAXOSMITHKLINE   (United States)

Author keywords

75Se homocholic acid taurine; Brush border membrane vesicles; CAS RN 178961 24 5; Cholesterol 7 monooxygenase; Human ileal apical sodium dependent bile acid co transporter; Hypocholesterolemic agents; Mice; Monkeys; Rats; Taurocholic acid

Indexed keywords

3 BUTYL 3 ETHYL 2,3,4,5 TETRAHYDRO 7,8 DIMETHOXY 5 PHENYL 1,4 BENZOTHIAZEPINE 1,1 DIOXIDE; BENZOTHIAZEPINE DERIVATIVE; BILE ACID; CHOLESTEROL; CHOLESTEROL 7ALPHA MONOOXYGENASE; LOW DENSITY LIPOPROTEIN; TAUROCHOLIC ACID; TAUROSELCHOLIC ACID SE 75; TRIACYLGLYCEROL; UNCLASSIFIED DRUG; VERY LOW DENSITY LIPOPROTEIN;

ANIMAL CELL; ANIMAL EXPERIMENT; APICAL MEMBRANE; ARTICLE; BILE ACID METABOLISM; BRUSH BORDER; CHO CELL; CHOLESTEROL METABOLISM; CIRCADIAN RHYTHM; CONTROLLED STUDY; DOSE RESPONSE; DRUG STRUCTURE; ENZYME ACTIVITY; ENZYME INDUCTION; HYPERCHOLESTEROLEMIA; MALE; MEMBRANE VESICLE; MONKEY; MOUSE; NONHUMAN; PRIORITY JOURNAL; RAT; SMALL INTESTINE;

EID: 0036692428     PISSN: 00222275     EISSN: None     Source Type: Journal    
DOI: 10.1194/jlr.m200121-jlr200     Document Type: Article

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