메뉴 건너뛰기




Volumn 22, Issue 1, 2002, Pages 29-35

Partial agonistic activity of labetalol, the arylethanolamine, on β3-adrenoceptors in the guinea-pig gastric fundus

Author keywords

[No Author keywords available]

Indexed keywords

4 (3 TERT BUTYLAMINO 2 HYDROXYPROPOXY) 2 BENZIMIDAZOLONE; 4 [2 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO]PROPYL]PHENOXYACETIC ACID; 4 [2 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO]PROPYL]PHENOXYACETIC ACID METHYL ESTER; ADRENALIN; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; ATENOLOL; BETA 3 ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR BLOCKING AGENT; BUPRANOLOL; BUTOXAMINE; ISOPRENALINE; LABETALOL; NORADRENALIN; PARTIAL AGONIST; ETHANOLAMINE;

EID: 0036479440     PISSN: 14748665     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1474-8673.2002.00239.x     Document Type: Article
Times cited : (3)

References (27)
  • 1
    • 0038191562 scopus 로고    scopus 로고
    • (1980). Ethanamine derivatives: their preparation and use in pharmacological compositions. European Patent, 02385
    • AINSWORTH, A.T. & SMITH, D.G. (1980). Ethanamine derivatives: their preparation and use in pharmacological compositions. European Patent, 02385.
    • Ainsworth, A.T.1    Smith, D.G.2
  • 4
    • 0025321911 scopus 로고
    • In vitro inhibition of intestinal motility by phenylethanolaminotetralines: Evidence of atypical β-adrenoceptors in rat colon
    • BIANCHETTI, A. & MANARA, L. (1990). In vitro inhibition of intestinal motility by phenylethanolaminotetralines: evidence of atypical β-adrenoceptors in rat colon. Br. J. Pharmacol., 100, 831-839.
    • (1990) Br. J. Pharmacol. , vol.100 , pp. 831-839
    • Bianchetti, A.1    Manara, L.2
  • 5
    • 0019985252 scopus 로고
    • The alpha- and beta-adrenoceptor blocking potencies of labetalol and its individual stereoisomers in anaesthetized dogs and in isolated tissues
    • BRITTAIN, R.T., DREW, G.M. & LEVY, G.P. (1982). The alpha- and beta-adrenoceptor blocking potencies of labetalol and its individual stereoisomers in anaesthetized dogs and in isolated tissues. Br. J. Pharmacol., 77, 105-114.
    • (1982) Br. J. Pharmacol. , vol.77 , pp. 105-114
    • Brittain, R.T.1    Drew, G.M.2    Levy, G.P.3
  • 6
    • 0017072055 scopus 로고
    • A review of the animal pharmacology of labetalol, a combined alpha- and beta-adrenoceptor-blocking drug
    • BRITTAIN, R.T. & LEVY, G.P. (1976). A review of the animal pharmacology of labetalol, a combined alpha- and beta-adrenoceptor-blocking drug. Br. J. Clin. Pharmacol., 3, 681-684.
    • (1976) Br. J. Clin. Pharmacol. , vol.3 , pp. 681-684
    • Brittain, R.T.1    Levy, G.P.2
  • 7
    • 0018294332 scopus 로고
    • β-adrenoceptor agonist activity of labetolol on the isolated uterus of the rat
    • CAREY, B. & WHALLEY, E.T. (1979a). β-Adrenoceptor agonist activity of labetolol on the isolated uterus of the rat. Br. J. Pharmacol., 67, 13-15.
    • (1979) Br. J. Pharmacol. , vol.67 , pp. 13-15
    • Carey, B.1    Whalley, E.T.2
  • 8
    • 0018712512 scopus 로고
    • Labetalol possesses β-adrenoceptor agonist action on the rat isolated uterus
    • CAREY, B. & WHALLEY, E.T. (1979b). Labetalol possesses β-adrenoceptor agonist action on the rat isolated uterus. J. Pharm. Pharmacol., 31, 791-792.
    • (1979) J. Pharm. Pharmacol. , vol.31 , pp. 791-792
    • Carey, B.1    Whalley, E.T.2
  • 9
    • 0019774401 scopus 로고
    • Intrinsic activity of labetalol on guinea-pig isolated trachea
    • CARPENTER, J.R. (1981). Intrinsic activity of labetalol on guinea-pig isolated trachea. J. Pharm. Pharmacol., 33, 806-807.
    • (1981) J. Pharm. Pharmacol. , vol.33 , pp. 806-807
    • Carpenter, J.R.1
  • 10
    • 0002638731 scopus 로고
    • β-adrenoceptors in guinea-pig gastric fundus - Are they the same as the 'atypical' β-adrenoceptors in rat adipocytes?
    • COLEMAN, R.A., DENYER, L.H. & SHELDRICK, K.E. (1987). β-Adrenoceptors in guinea-pig gastric fundus - are they the same as the 'atypical' β-adrenoceptors in rat adipocytes? Br. J. Pharmacol., 90, 40P.
    • (1987) Br. J. Pharmacol. , vol.90
    • Coleman, R.A.1    Denyer, L.H.2    Sheldrick, K.E.3
  • 11
    • 0015376880 scopus 로고
    • Pharmacology of AH 5158; a drug which blocks both α- and β-adrenoceptors
    • FARMER, J.B., KENNEDY, I., LEVY, G.P. & MARSHALL, R.J. (1972). Pharmacology of AH 5158; a drug which blocks both α- and β-adrenoceptors. Br. J. Pharmacol., 45, 660-675.
    • (1972) Br. J. Pharmacol. , vol.45 , pp. 660-675
    • Farmer, J.B.1    Kennedy, I.2    Levy, G.P.3    Marshall, R.J.4
  • 12
    • 0032709043 scopus 로고    scopus 로고
    • 3-adrenoceptor antagonist bupranolol
    • 3-adrenoceptor antagonist bupranolol. Pharmacology, 59, 290-297.
    • (1999) Pharmacology , vol.59 , pp. 290-297
    • Horinouchi, T.1    Koike, K.2
  • 13
    • 0033033880 scopus 로고    scopus 로고
    • Characterization of atypical β-adrenoceptors in the guinea-pig duodenum
    • HORINOUCHI, T. & KOIKE, K. (1999b). Characterization of atypical β-adrenoceptors in the guinea-pig duodenum. Eur. J. Pharmacol., 376, 61-66.
    • (1999) Eur. J. Pharmacol. , vol.376 , pp. 61-66
    • Horinouchi, T.1    Koike, K.2
  • 14
    • 0034284270 scopus 로고    scopus 로고
    • Partial agonist activity of carteolol on atypical β-adrenoceptors in the guinea-pig duodenum
    • HORINOUCHI, T. & KOIKE, K. (2000a). Partial agonist activity of carteolol on atypical β-adrenoceptors in the guinea-pig duodenum. Eur. J. Pharmacol., 403, 133-138.
    • (2000) Eur. J. Pharmacol. , vol.403 , pp. 133-138
    • Horinouchi, T.1    Koike, K.2
  • 15
    • 0034528098 scopus 로고    scopus 로고
    • Partial agonistic effects of carteolol on atypical β-adrenoceptors in the guinea-pig gastric fundus
    • HORINOUCHI, T. & KOIKE, K. (2000b). Partial agonistic effects of carteolol on atypical β-adrenoceptors in the guinea-pig gastric fundus. Jpn. J. Pharmacol., 84, 287-292.
    • (2000) Jpn. J. Pharmacol. , vol.84 , pp. 287-292
    • Horinouchi, T.1    Koike, K.2
  • 16
    • 0035937456 scopus 로고    scopus 로고
    • Functional properties of atypical β-adrenoceptors on the guinea-pig duodenum
    • HORINOUCHI, T. & KOIKE, K. (2001a). Functional properties of atypical β-adrenoceptors on the guinea-pig duodenum. Eur. J. Pharmacol., 416, 153-163.
    • (2001) Eur. J. Pharmacol. , vol.416 , pp. 153-163
    • Horinouchi, T.1    Koike, K.2
  • 17
    • 0034746225 scopus 로고    scopus 로고
    • (±)-Pindolol acts as a partial agonist at atypical β-adrenoceptors in the guinea-pig duodenum
    • HORINOUCHI, T. & KOIKE, K. (2001b). (±)-Pindolol acts as a partial agonist at atypical β-adrenoceptors in the guinea-pig duodenum. Jpn. J. Pharmacol., 85, 35-40.
    • (2001) Jpn. J. Pharmacol. , vol.85 , pp. 35-40
    • Horinouchi, T.1    Koike, K.2
  • 18
    • 0030030731 scopus 로고    scopus 로고
    • (-)-CGP 12177-induced increase of human atrial contraction through a putative third β-adrenoceptor
    • KAUMANN, A.J. (1996). (-)-CGP 12177-induced increase of human atrial contraction through a putative third β-adrenoceptor. Br. J. Pharmacol., 117, 93-98.
    • (1996) Br. J. Pharmacol. , vol.117 , pp. 93-98
    • Kaumann, A.J.1
  • 20
    • 0028978560 scopus 로고
    • Possible mechanisms of β-adrenoceptor-mediated relaxation induced by noradrenaline in guinea-pig taenia caecum
    • KOIKE, K., HORINOUCHI, T. & TAKAYANAGI, I. (1995). Possible mechanisms of β-adrenoceptor-mediated relaxation induced by noradrenaline in guinea-pig taenia caecum. Eur. J. Pharmacol., 279, 159-163.
    • (1995) Eur. J. Pharmacol. , vol.279 , pp. 159-163
    • Koike, K.1    Horinouchi, T.2    Takayanagi, I.3
  • 24
    • 0018655874 scopus 로고
    • 2 and receptor differentiation: A statistical analysis of competitive antagonism
    • 2 and receptor differentiation: a statistical analysis of competitive antagonism. Life Sci., 25, 637-654.
    • (1979) Life Sci. , vol.25 , pp. 637-654
    • Tallarida, R.J.1    Cowan, A.2    Adler, M.W.3
  • 25
    • 73649209211 scopus 로고
    • Cumulative dose-response curves, II. Technique for the making of dose-response curves in isolated organs and the evaluation of drug parameters
    • VAN ROSSUM, J.M. (1963). Cumulative dose-response curves, II. Technique for the making of dose-response curves in isolated organs and the evaluation of drug parameters. Arch. Int. Pharmacodyn., 143, 299-330.
    • (1963) Arch. Int. Pharmacodyn. , vol.143 , pp. 299-330
    • Van Rossum, J.M.1
  • 26
    • 0017754150 scopus 로고
    • The cardiovascular and uterine effects of labetolol in conscious normotensive pregnant rats
    • WHALLEY, E.T. (1977). The cardiovascular and uterine effects of labetolol in conscious normotensive pregnant rats. Br. J. Pharmacol., 61, 505P-506P.
    • (1977) Br. J. Pharmacol. , vol.61 , pp. 505-506
    • Whalley, E.T.1
  • 27
    • 0018897783 scopus 로고
    • Observations on the effect of labetalol on pregnancy and parturition in normotensive rats
    • WHALLEY, E.T. (1980). Observations on the effect of labetalol on pregnancy and parturition in normotensive rats. Gen. Pharmacol., 11, 297-302.
    • (1980) Gen. Pharmacol. , vol.11 , pp. 297-302
    • Whalley, E.T.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.