The selectivity in vitro of the stereoisomers of the beta-3 adrenoceptor agonist BRL 37344

Journal of Pharmacology and Experimental Therapeutics

Volumn 277, Issue 1, 1996, Pages 22-27

  Oriowo, M Ayo ^a,b   Chapman, Helen ^a   Kirkham, David M ^a,c   Sennitt, Matthew V ^a,d   Ruffolo Jr , Robert R ^a   Cawthorne, Michael A ^a,e  

^a GLAXOSMITHKLINE   (United Kingdom)

^b KUWAIT UNIVERSITY   (Kuwait)

^c UNIVERSITY OF BIRMINGHAM   (United Kingdom)

^d ST GEORGE S HOSPITAL   (United Kingdom)

^e UNIVERSITY OF BUCKINGHAM   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

4 [2 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO]PROPYL]PHENOXYACETIC ACID; BETA 3 ADRENERGIC RECEPTOR STIMULATING AGENT; RECEPTOR SUBTYPE;

ADIPOCYTE; ADIPOSE TISSUE; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BETA ADRENERGIC STIMULATION; DRUG POTENCY; DRUG SELECTIVITY; ENANTIOMER; FEMALE; LIPOLYSIS; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; RECEPTOR UPREGULATION; STEREOCHEMISTRY; UTERUS RELAXATION;

ADRENERGIC BETA-AGONISTS; ANIMALS; DOSE-RESPONSE RELATIONSHIP, DRUG; ETHANOLAMINES; FEMALE; HEART RATE; MALE; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, ADRENERGIC, BETA; RECEPTORS, ADRENERGIC, BETA-3; STEREOISOMERISM; UTERINE CONTRACTION;

EID: 0030439764     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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