Potent and selective partial ecdysone agonist activity of chromafenozide in Sf9 cells

Biochemical and Biophysical Research Communications

Volumn 292, Issue 4, 2002, Pages 1087-1091

  Toya, Tetsuya ^a   Masui, Akio ^a   Fukasawa, Hiroshi ^b   Endo, Yasuyuki ^b  

^a NIPPON KAYAKU CO LTD   (Japan)

^b UNIVERSITY OF TOKYO   (Japan)

Author keywords

Agonist; ANS 118; Assay; Chromafenozide; Ecdysone; Insect hormone; Kc cells; Luciferase; Ponasterone A; Sf9 cells

Indexed keywords

CHROMAFENOZIDE; ECDYSONE; ECDYSONE RECEPTOR; ECDYSTERONE; HORMONE RECEPTOR; PONASTERONE A; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DOSE RESPONSE; GENETIC TRANSCRIPTION; HORMONE ACTION; LEPIDOPTERA; MOLTING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; REPORTER GENE;

INSECTA; LEPIDOPTERA;

EID: 0036295599     PISSN: 0006291X     EISSN: None     Source Type: Journal    
DOI: 10.1006/bbrc.2002.6771     Document Type: Article

References (19)

1. Juvenile hormone: The status of its "status quo" action
2. Recent advances in our knowledge of ecdysteroid biosynthesis in insects and crustaceans
3. The Drosophila EcR gene encodes an ecdysone receptor, a new member of the steroid receptor superfamily
4. The RXR heterodimers and orphan Receptors
5. The nuclear receptor superfamily: The second decade
6. Ecdysone receptors and their biological actions
7. Functional ecdysone receptor is the product of EcR and ultraspiracle genes
8. Dueling orphans: Interacting nuclear receptors coordinate Drosophila metamorphosis
9. RH 5849, a nonsteroidal ecdysone agonist: Effects on a Drosophila cell line
10. RH 5849, a nonsteroidal ecdysone agonist: Effects on laval lepidoptera
11. Field evaluation of RH 5992 on Lepidopterous pests in Europe
12. ANS-118 a novel insecticide
13. Synthesis and insecticidal activity of benzoheterocyclic analogues of dibenzoylhydrazine. Part 3: Mod-ification of the hydrazine part
14. An automated ecdysteroid receptor binding assay using a 96-well microplate
15. Bombyx mori (BmEcR) and Bombyx USP (BmCF1) combine to form a functional ecdysone receptor
16. Expression of EcR and USP in Escherichia coli: Purification and functional studies
17. Sensitive, rapid and simple method for evaluation of ecdysteroid agonist activity based on the mode of action of the hormone
18. Structure-activity study and conformational analysis of RH-5992, the first commercialized nonsteroidal ecdysone agonist
19. A new model for 20-hydroxyecdysone and dibenzoylhydrazine binding: A homology modeling and docking approach