Quantitative structure activity relationships for the glucuronidation of simple phenols by expressed human UGT1A6 and UGT1A9

Drug Metabolism and Disposition

Volumn 30, Issue 6, 2002, Pages 734-738

  Ethell, Brian T ^a   Ekins, Sean ^b   Wang, Jibo ^b   Burchell, Brian ^a  

^a UNIVERSITY OF DUNDEE   (United Kingdom)

^b ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PHENOL DERIVATIVE;

ARTICLE; CONTROLLED STUDY; DRUG GLUCURONIDATION; ENZYME ACTIVITY; ENZYME KINETICS; HUMAN; HUMAN CELL; HUMAN TISSUE; MOLECULAR DYNAMICS; MOLECULAR MODEL; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN EXPRESSION; QUANTITATIVE STRUCTURE ACTIVITY RELATION; VALIDATION PROCESS;

CELL LINE; GLUCURONIDES; GLUCURONOSYLTRANSFERASE; HUMANS; ISOENZYMES; KINETICS; MOLECULAR STRUCTURE; PHENOLS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0036266180     PISSN: 00909556     EISSN: None     Source Type: Journal    
DOI: 10.1124/dmd.30.6.734     Document Type: Article

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