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Journal of Pharmacology and Experimental Therapeutics

Volumn 300, Issue 2, 2002, Pages 577-582

Pharmacological characterization of SC-57461A (3-[methyl[3-[4-(phenylmethyl)phenoxy]propyl]amino]propanoic acid HCl), a potent and selective inhibitor of leukotriene A4 hydrolase I: In vitro studies

(6) Askonas, Leslie J a Kachur, James F a Villani Price, Doreen a Liang, Chi Dean D a Russell, Mark A a Smith, Walter G a

a PFIZER INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3 [METHYL [3 [4 (PHENYLMETHYL)PHENOXY]PROPYL]AMINO]PROPANOIC ACID; LEUKOTRIENE A4 HYDROLASE; LEUKOTRIENE B4; LEUKOTRIENE RECEPTOR BLOCKING AGENT; SC 57461A; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; DRUG INHIBITION; DRUG MECHANISM; DRUG STRUCTURE; ENTERITIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; MOUSE; NONHUMAN; PATHOGENESIS; PRIORITY JOURNAL; PSORIASIS; RAT;

AMINOPEPTIDASES; ANIMALS; ARACHIDONIC ACID; BETA-ALANINE; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DOGS; EICOSANOIDS; ENZYME INHIBITORS; ENZYME-LINKED IMMUNOSORBENT ASSAY; EPOXIDE HYDROLASES; HUMANS; IONOPHORES; KINETICS; LEUKOTRIENE A4; LEUKOTRIENE ANTAGONISTS; MACACA MULATTA; MICE; RATS; RECOMBINANT PROTEINS; SPECIES SPECIFICITY; SUBSTRATE SPECIFICITY;

EID: 0036154531 PISSN: 00223565 EISSN: None Source Type: Journal
DOI: 10.1124/jpet.300.2.577 Document Type: Article

Times cited : (37)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.