The motilin pharmacophore in CHO cells expressing the human motilin receptor

Biochemical and Biophysical Research Communications

Volumn 293, Issue 4, 2002, Pages 1223-1227

  Thielemans, Leen ^a   Depoortere, Inge ^a   Vanden Broeck, Jozef ^a   Peeters, Theo L ^a  

^a UNIVERSITY OF LEUVEN   (Belgium)

Author keywords

Aequorin; Calcium; CHO cell; Luminescence; Motilin; Pharmacophore; Receptor

Indexed keywords

ALANINE; CALCIUM ION; ERYTHROMYCIN; ERYTHROMYCIN A ENOL ETHER; ERYTHROMYCIN B ENOL ETHER; MACROLIDE; MOTILIN; MOTILIN DERIVATIVE; MOTILIN[1 ALANINE 13 LEUCINE]; MOTILIN[10 ALANINE 13 LEUCINE]; MOTILIN[11 ALANINE 13 LEUCINE]; MOTILIN[12 ALANINE 13 LEUCINE]; MOTILIN[13 ALANINE 13 LEUCINE]; MOTILIN[13 LEUCINE]; MOTILIN[2 ALANINE 13 LEUCINE]; MOTILIN[3 ALANINE 13 LEUCINE]; MOTILIN[4 ALANINE 13 LEUCINE]; MOTILIN[5 ALANINE 13 LEUCINE]; MOTILIN[6 ALANINE 13 LEUCINE]; MOTILIN[7 ALANINE 13 LEUCINE]; MOTILIN[8 ALANINE 13 LEUCINE]; MOTILIN[9 ALANINE 13 LEUCINE]; N ETHYL N METHYL ERYTHROMYCIN A; N ETHYL N METHYL ERYTHROMYCIN A ENOL ETHER; PHENYLALANINE; RECEPTOR PROTEIN; TYROSINE; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; AMINO TERMINAL SEQUENCE; ARTICLE; CALCIUM TRANSPORT; CELL MEMBRANE TRANSPORT; CHO CELL; CONTROLLED STUDY; CORRELATION ANALYSIS; DRUG EFFECT; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; HUMAN; HUMAN CELL; NONHUMAN; PHARMACOPHORE; PRIORITY JOURNAL; PROTEIN CONFORMATION; PROTEIN EXPRESSION; PROTEIN FUNCTION; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

AEQUORIN; ALANINE; ANIMALS; CALCIUM; CHO CELLS; CRICETINAE; DIGESTIVE SYSTEM; DUODENUM; ERYTHROMYCIN; GASTROINTESTINAL AGENTS; HUMANS; MOTILIN; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; RABBITS; RECEPTORS, GASTROINTESTINAL HORMONE; RECEPTORS, NEUROPEPTIDE; STRUCTURE-ACTIVITY RELATIONSHIP; SWINE; THYROID GLAND;

ORYCTOLAGUS CUNICULUS;

EID: 0036072904     PISSN: 0006291X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-291X(02)00356-X     Document Type: Article

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