The pure anti-oestrogen ICI 182,780 (Faslodex™) activates large conductance Ca 2+-activated K + channels in smooth muscle

British Journal of Pharmacology

Volumn 136, Issue 7, 2002, Pages 961-964

  Dick, Gregory M ^a  

^a UNIVERSITY OF NEVADA SCHOOL OF MEDICINE   (United States)

Author keywords

1 subunit; 17 Oestradiol; MaxiK channel; Slo; Tamoxifen

Indexed keywords

ANTIESTROGEN; CALCIUM CHANNEL; CELL NUCLEUS RECEPTOR; ESTROGEN; ESTROGEN RECEPTOR; FULVESTRANT; POTASSIUM CHANNEL; TAMOXIFEN; CALCIUM ACTIVATED POTASSIUM CHANNEL; DRUG DERIVATIVE; ESTRADIOL;

ANIMAL CELL; ARTICLE; BINDING SITE; CONTROLLED STUDY; HYPOTHESIS; INTESTINE MUSCLE; MEMBRANE BINDING; MUSCLE CELL; NONHUMAN; PRIORITY JOURNAL; PROBABILITY; SMOOTH MUSCLE; ANIMAL; CHANNEL GATING; COLON; COMPARATIVE STUDY; CYTOLOGY; DOG; DRUG EFFECT; IN VITRO STUDY; METABOLISM; PATCH CLAMP; PHYSIOLOGY;

ANIMAL; COLON; COMPARATIVE STUDY; DOGS; ESTRADIOL; ESTROGEN ANTAGONISTS; IN VITRO; ION CHANNEL GATING; MUSCLE CELLS; MUSCLE, SMOOTH; PATCH-CLAMP TECHNIQUES; POTASSIUM CHANNELS, CALCIUM-ACTIVATED; SUPPORT, U.S. GOV'T, P.H.S.; TAMOXIFEN; ANIMALS;

EID: 0036024230     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0704807     Document Type: Article

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