Transbuccal peptide delivery: Stability and in vitro permeation studies on endomorphin-1

Journal of Controlled Release

Volumn 73, Issue 1, 2001, Pages 31-36

  Bird, Aaron P ^a   Faltinek, Jennifer R ^a   Shojaei, Amir H ^b  

^a TEXAS TECH UNIVERSITY HEALTH SCIENCES CENTER   (United States)

^b Shire Laboratories Inc   (United States)

Author keywords

Buccal mucosa; Diprotin A; Endomorphin 1; Peptide delivery; Peptide stability; Transbuccal delivery

Indexed keywords

BUFFER; DIPEPTIDYL PEPTIDASE IV; DIPROTIN A; ENDOMORPHIN 1; GLYCOCHOLATE SODIUM; MU OPIATE RECEPTOR; MU OPIATE RECEPTOR AGONIST; RECEPTOR SUBTYPE; TAUROCHOLIC ACID;

ANIMAL TISSUE; ARTICLE; CHEEK MUCOSA; CONTROLLED DRUG RELEASE; CONTROLLED STUDY; DEGRADATION; DRUG DEGRADATION; DRUG DELIVERY SYSTEM; DRUG PENETRATION; DRUG POTENCY; DRUG SELECTIVITY; DRUG SPECIFICITY; DRUG STABILITY; ENZYME INHIBITION; ENZYME ISOLATION; NONHUMAN; PH; PRIORITY JOURNAL; SWINE;

ADMINISTRATION, BUCCAL; ALGORITHMS; ANALGESICS, OPIOID; ANIMALS; BUFFERS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DRUG DELIVERY SYSTEMS; DRUG STABILITY; ENDOPEPTIDASES; MOUTH MUCOSA; OLIGOPEPTIDES; PERMEABILITY; PROTEASE INHIBITORS; SOLUTIONS; SWINE;

EID: 0035907175     PISSN: 01683659     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0168-3659(01)00246-2     Document Type: Article

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