Nucleosides and nucleotides. 200. Reinvestigation of 5′-N-ethylcarboxamidoadenosine derivatives: Structure-activity relationships for P3 purinoceptor-like proteins

Journal of Medicinal Chemistry

Volumn 44, Issue 2, 2001, Pages 208-214

  Umino, T ^a   Yoshioka, K ^b   Saitoh, Y ^b   Minakawa, N ^a   Nakata, H ^b   Matsuda, A ^a  

^a HOKKAIDO UNIVERSITY   (Japan)

^b TOKYO METROPOLITAN INSTITUTE OF MEDICAL SCIENCE   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

1 (ADENIN 9 YL) 1 DEOXY N CYCLOHEXYL BETA DEXTRO RIBOFURANURONAMIDE; 1 (ADENIN 9 YL) 1 DEOXY N ETHYL BETA DEXTRO RIBOFURANURONAMIDE; 1 (ADENIN 9 YL) 1 DEOXY N N PENTYL BETA DEXTRO RIBOFURANURONAMIDE; 9 (6,7 DIDEOXY BETA DEXTRO ALLOHEPT 5 YNOFURANOSYL)ADENINE; ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A1 RECEPTOR; ADENOSINE A2A RECEPTOR; ADENOSINE A2B RECEPTOR; ADENOSINE A3 RECEPTOR; ADENOSINE RECEPTOR; ALKYL GROUP; AMIDE; BINDING PROTEIN; HAK 2701; LIGAND; NITROGEN; NUCLEOSIDE; NUCLEOTIDE; P3 PURINORECEPTOR LIKE PROTEIN; PURINE P2 RECEPTOR; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; HYDROPHOBICITY; LIGAND BINDING; MUSCLE RELAXATION; RABBIT; STRUCTURE ACTIVITY RELATION; THORACIC AORTA;

ADENOSINE; ANIMALS; BRAIN; LIGANDS; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; RADIOLIGAND ASSAY; RATS; RECEPTORS, PURINERGIC; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035905865     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm000150k     Document Type: Article

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