Characterisation of agonist binding on human 5-HT2C receptor isoforms

European Journal of Pharmacology

Volumn 419, Issue 2-3, 2001, Pages 107-112

  Quirk, Kathleen ^a   Lawrence, Anthony ^a   Jones, Julie ^a   Misra, Anil ^a   Harvey, Victoria ^a   Lamb, Helen ^a   Revell, Dean ^a   Porter, Richard H P ^a   Knight, Antony R ^a  

^a Vernalis PLC   (United Kingdom)

Author keywords

5 HT (5 hydroxytryptamine, serotonin); 5 HT2C receptor INI; 5 HT2C receptor VSV; G protein; Isoform

Indexed keywords

(3 CHLOROPHENYL)PIPERAZINE; 1 (3 TRIFLUOROMETHYLPHENYL)PIPERAZINE; 2 (6 CHLORO 5 FLUORO 1 INDOLYL) 1 METHYLETHYLAMINE; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 4 IODO 2,5 DIMETHOXYAMPHETAMINE; 6 CHLORO 2 (1 PIPERAZINYL)PYRAZINE; BROLAMFETAMINE; GUANINE NUCLEOTIDE BINDING PROTEIN; ISOPROTEIN; KETANSERIN; MESULERGINE; SEROTONIN; SEROTONIN 2C RECEPTOR;

AGONIST; ANIMAL CELL; ARTICLE; BINDING SITE; CHO CELL; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; HUMAN; HUMAN CELL; KIDNEY CELL; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; RNA EDITING;

ANIMALS; BINDING SITES; CHO CELLS; CRICETINAE; GTP-BINDING PROTEINS; HUMANS; PROTEIN ISOFORMS; RECEPTOR, SEROTONIN, 5-HT2C; RECEPTORS, SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS;

EID: 0035843751     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(01)00943-8     Document Type: Article

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