Tandem Michael addition - Hoffman elimination sequence of DMAD on tetrahydropyrrolo[3,2-c]pyridines. New route to vinylpyrroles

Heterocyclic Communications

Volumn 7, Issue 5, 2001, Pages 461-466

  Varlamov, Alexey V ^a   Borisova, Tatiana N ^a   Voskressensky, Leonid G ^a   Nsabimana, Bonifas ^a   Chernyshev, Alexey I ^a  

^a PEOPLES FRIENDSHIP UNIVERSITY OF RUSSIA   (Russian Federation)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0035733072     PISSN: 07930283     EISSN: None     Source Type: Journal    
DOI: 10.1515/HC.2001.7.5.461     Document Type: Article

References (8)

1. A.C. Cope, A.R. Trumbull, Org.React., 11,317(1960).
2. J. Braun von, Ber., 37, 2915(1904)
3. A.V. Varlamov, T.N. Borisova, L.G. Voskressensky, A.A. Brook, A.I. Chernyhev, ARKIVOC, 1, 2, 159-162, (2000).
4. C. Altomare, L. Summo, S. Cellamare, A.V. Varlamov, L..G. Voskressensky, T.N. Borisova, A. Carroti, Bioorg. Med.Chem.Lett., 10, 581, (2000).
5. K. Nozaki, N. Sato, K. Ikeda, H. Takaya, J Org Chem, 61, 14, 4516, (1996).
6. R.A. Jones In Pyrroles, John Wiley & Sons Inc.: New York, 1990; Part II.
7. For pyrrolo[3,2-c]piperidines synthesis via piperidones oximes heterocyclization with acetylene (Trofimov reaction) see: (a) T. N. Borisova, A. V. Varlamov, N. D. Sergeeva, A. T. Soldatenkov, O. V. Zvolinskii, Chem.Heterocycl.Compd.(Engl.Transl.), 23, 7, 799, (1987). For a review of Trofimov reaction see (b) B. A. Trofimov, A. I. Mikhaleva, Heterocycles, 37, 2, 1193, (1994).
8. For pyrrolo[3,2-c]piperidines synthesis via piperidones oximes heterocyclization with acetylene (Trofimov reaction) see: (a) T. N. Borisova, A. V. Varlamov, N. D. Sergeeva, A. T. Soldatenkov, O. V. Zvolinskii, Chem.Heterocycl.Compd.(Engl.Transl.), 23, 7, 799, (1987). For a review of Trofimov reaction see (b) B. A. Trofimov, A. I. Mikhaleva, Heterocycles, 37, 2, 1193, (1994).