Evaluation of the conformational propensities of peptide isosteres as a basis for selecting bioactive pseudopeptides

Journal of Peptide Research

Volumn 58, Issue 6, 2001, Pages 546-561

  Gupta, S ^a   Payne, J W ^a  

^a BANGOR UNIVERSITY   (United Kingdom)

Author keywords

Conformational analysis; Conformational entropy; Drug delivery; Drug design; Ligand binding; Molecular modelling; Peptide conformers; Peptide transport

Indexed keywords

AMPHOLYTE; CARRIER PROTEIN; DIPEPTIDE; N METHYLAMIDE; PSEUDOPEPTIDE; RETROAMIDE; THIOAMIDE; TRIPEPTIDE; UNCLASSIFIED DRUG;

ARTICLE; CONFORMATIONAL TRANSITION; MOLECULAR RECOGNITION; PEPTIDE ANALYSIS; PRIORITY JOURNAL; PROTEIN CONFORMATION; STRUCTURE ANALYSIS;

DIPEPTIDES; DRUG DESIGN; MODELS, MOLECULAR; MOLECULAR MIMICRY; OLIGOPEPTIDES; PEPTIDES; PROTEIN CONFORMATION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035717847     PISSN: 1397002X     EISSN: None     Source Type: Journal    
DOI: 10.1034/j.1399-3011.2001.00954.x     Document Type: Article

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