A new ring-forming methodology for the synthesis of conformationally constrained bioactive molecules

Chemistry Letters

Volumn , Issue 3, 2001, Pages 192-193

  Papahatjis, Demetris P ^c   Nikas, Spyros ^c   Tsotinis, Andrew ^a   Vlachou, Margarita ^a   Makriyannis, Alexandros ^b  

^a UNIVERSITY OF ATHENS   (Greece)

^b UNIVERSITY OF CONNECTICUT   (United States)

^c INSTITUTE OF BIOLOGY   (Greece)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0035649958     PISSN: 03667022     EISSN: None     Source Type: Journal    
DOI: 10.1246/cl.2001.192     Document Type: Article

References (10)

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9. Use of potassium bis(trimethylsilyl)amide (5 equiv) and 1,2-dichloroethane (3 equiv) was found to be more effective (68% yield).
10. Use of potassium bis(trimethylsilyl)amide (5 equiv) and 1,2-dichloroethane (3 equiv) was found to be more effective (62% yield).