Regulation of agonist binding to rat ETB receptors by cations and GTPγS

Biochemical Pharmacology

Volumn 62, Issue 5, 2001, Pages 537-545

  Ceccarelli, Francesca ^a   Giusti, Laura ^a   Bigini, Gianni ^a   Costa, Barbara ^a   Grillotti, Dante ^a   Fiumalbi, Erika ^a   Lucacchini, Antonio ^a   Mazzoni, Maria Rosa ^a  

^a UNIVERSITY OF PISA   (Italy)

Author keywords

Cations; Endothelin receptors; Endothelins; ETB receptor; G protein coupled receptors; Heterotrimeric G proteins

Indexed keywords

DIVALENT CATION; ENDOTHELIN 1; ENDOTHELIN 3; ENDOTHELIN B RECEPTOR; GUANOSINE 5' O (2 THIODIPHOSPHATE); IODINE 125; MAGNESIUM CHLORIDE; MAGNESIUM ION; MONOVALENT CATION; N (2,6 DIMETHYLPIPERIDINOCARBONYL) 4 METHYLLEUCYL DEXTRO (1 METHOXYCARBONYLTRYPTOPHANYL) DEXTRO NORLEUCINE; RECEPTOR SUBTYPE; SODIUM CHLORIDE; SODIUM ION; SUCCINYLENDOTHELIN 1 [8-21][9 GLUTAMIC ACID 11,15 ALANINE];

ANIMAL TISSUE; ARTICLE; CEREBELLUM; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG MECHANISM; MALE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR BINDING; RECEPTOR UPREGULATION;

ANIMALS; BINDING, COMPETITIVE; CATIONS; ENDOTHELIN-3; ENDOTHELINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); IODINE RADIOISOTOPES; MAGNESIUM; MALE; PEPTIDE FRAGMENTS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTOR, ENDOTHELIN B; RECEPTORS, ENDOTHELIN; SODIUM;

EID: 0035452132     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(01)00706-7     Document Type: Article

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