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Volumn 36, Issue 5, 2001, Pages 447-460

Stereospecific synthesis and biological evaluations of β-L-pentofuranonucleoside derivatives of 5-fluorouracil and 5-fluorocytosine

(8) Griffon, Jean François a Mathé, Christophe a Faraj, Abdesslem b Aubertin, Anne Marie c De Clercq, Erik d Balzarini, Jan d Sommadossi, Jean Pierre e Gosselin, Gilles a,b

a UNIVERSITÉ DE MONTPELLIER (France)

b CNRS (France)

c UNIVERSITÉ DE STRASBOURG (France)

d REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

e Novirio Pharmaceuticals (United States)

Author keywords

L nucleoside analogues; 5 Fluorocytosine; 5 Fluorouracil; Anti HBV activity; Anti HIV activity; Anti tumoral activity

Indexed keywords

1 (2 DEOXY BETA LEVO ERYTHRO PENTOFURANOSYL) 5 FLUOROCYTOSIN; 1 (2 DEOXY BETA LEVO ERYTHRO PENTOFURANOSYL) 5 FLUOROURACIL; 1 (2 DEOXY BETA LEVO THREO PENTOFURANOSYL) 5 FLUOROCYTOSINE; 1 (2 DEOXY BETA LEVO THREO PENTOFURANOSYL) 5 FLUOROURACIL; 1 (BETA LEVO ARABINOFURANOSYL) 5 FLUOROCYTOSINE; 1 (BETA LEVO ARABINOFURANOSYL) 5 FLUOROURACIL; 1 (BETA LEVO RIBOFURANOSYL) 5 FLUOROCYTOSINE; 1 (BETA LEVO RIBOFURANOSYL) 5 FLUOROURACIL; 1 (BETA LEVO XYLOFURANOSYL) 5 FLUOROCYTOSINE; 1 (BETA LEXO XYLOFURANOSYL) 5 FLUOROURACIL; 2' DEOXY BETA DEXTRO RIBOFURANONUCLEOSIDE 5 FLUORORACIL; ANTIINFECTIVE AGENT; ANTIVIRUS AGENT; BETA LEVO PENTOFURANONUCLEOSIDE DERIVATIVE; FLUCYTOSINE; FLUCYTOSINE DERIVATIVE; FLUOROURACIL DERIVATIVE; NUCLEOSIDE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL MODEL; ANTIVIRAL ACTIVITY; ARTICLE; BREAST CARCINOMA; CANCER INHIBITION; CONTROLLED STUDY; DRUG EFFECT; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HEPATITIS; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; LEUKEMIA; MOUSE; NONHUMAN; REACTION ANALYSIS; STEREOSPECIFICITY; T LYMPHOCYTE; TUMOR CELL;

ANIMALS; ANTI-HIV AGENTS; ANTINEOPLASTIC AGENTS; CELL DIVISION; DRUG DESIGN; FLUCYTOSINE; FLUOROURACIL; HIV; HUMANS; MICE; NUCLEOSIDES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; T-LYMPHOCYTES; TUMOR CELLS, CULTURED;

EID: 0035328957 PISSN: 02235234 EISSN: None Source Type: Journal
DOI: 10.1016/S0223-5234(01)01238-7 Document Type: Article

Times cited : (15)

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