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Volumn 36, Issue 3, 2001, Pages 255-264

Imidazo[1,2-a]quinoxalines: Synthesis and cyclic nucleotide phosphodiesterase inhibitory activity

(14) Parra, Stéphanie a Laurent, Florence b Subra, Guy a Deleuze Masquefa, Carine a Benezech, Veronique a Fabreguettes, Jean Roch a Vidal, Jean Pierre b Pocock, Tristan c Elliott, Keith c Small, Roger c Escale, Roger a Michel, Alain b Chapat, Jean Pierre a Bonnet, Pierre Antoine a

a Laboratoire de Pharmacochimie (France)

b UNIV MONTPELLIER (France)

c UNIVERSITY OF MANCHESTER (United Kingdom)

Author keywords

Halogen metal exchange; Imidazo 1,2 a quinoxaline; Lithiation; Phosphodiesterase inhibition; Smooth muscle relaxant activity

Indexed keywords

1 BROMO 4 METHOXYIMIDAZO[1,2 A]QUINOXALINE; 4 (METHYLAMINO)IMIDAZO[1,2 A]QUINOXALINE 2 CARBONITRILE; 5 (4 ACETAMIDOPHENYL) 2(1H) PYRAZINONE; 6 BROMO 8 METHYLAMINOIMIDAZO[1,2 A]PYRAZINE 2 CARBONITRILE; CYCLIC NUCLEOTIDE PHOSPHODIESTERASE; PHOSPHODIESTERASE INHIBITOR; QUINOXALINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CHEMICAL REACTION; CONTROLLED STUDY; CYCLIZATION; DRUG POTENCY; DRUG STRUCTURE; ENZYME INHIBITION; GUINEA PIG; MALE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; POLYMERIZATION; STRUCTURE ACTIVITY RELATION;

2',3'-CYCLIC-NUCLEOTIDE PHOSPHODIESTERASES; ANIMALS; CARDIOTONIC AGENTS; CATTLE; ENZYME INHIBITORS; GUINEA PIGS; INHIBITORY CONCENTRATION 50; ISOENZYMES; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MUSCLE RELAXATION; MUSCLE, SMOOTH; NITRILES; PYRAZINES; QUINOXALINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035310802 PISSN: 02235234 EISSN: None Source Type: Journal
DOI: 10.1016/S0223-5234(01)01213-2 Document Type: Article

Times cited : (30)

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