Allosteric modulation of the human 5-HT7A receptor by lipidic amphipathic compounds

Molecular Pharmacology

Volumn 60, Issue 6, 2001, Pages 1349-1355

  Alberts, G L ^a   Chio, C L ^a   Im, W B ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3 [(3 CHOLAMIDOPROPYL)DIMETHYLAMMONIO] 1 PROPANESULFONIC ACID; 5 CARBOXAMIDOTRYPTAMINE MALEATE; ADENYLATE CYCLASE; AMPHOPHILE; ARACHIDONIC ACID; BOVINE SERUM ALBUMIN; CYCLIC AMP; DOPAMINE 1 RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); GUANYLYLIMIDODIPHOSPHATE; LIPID; LISURIDE; LYSOPHOSPHATIDYLCHOLINE; LYSOPHOSPHOLIPID; MESULERGINE; METERGOLINE; METITEPINE; OLEIC ACID; PALMITIC ACID; SEROTONIN; SEROTONIN 1C RECEPTOR; SEROTONIN 1D RECEPTOR; SEROTONIN 7 RECEPTOR; SEROTONIN 7A RECEPTOR; SEROTONIN AGONIST; STEARIC ACID; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; BINDING AFFINITY; CONCENTRATION RESPONSE; HUMAN; HUMAN CELL; LIGAND BINDING; MODULATION; PRIORITY JOURNAL; RECEPTOR BINDING;

EID: 0035210810     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.60.6.1349     Document Type: Article

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