Colon-specific prodrugs of 5-aminosalicylic acid: Synthesis and in vitro/in vivo properties of acidic amino acid derivatives of 5-aminosalicylic acid

Journal of Pharmaceutical Sciences

Volumn 90, Issue 11, 2001, Pages 1767-1775

  Jung, Yun Jin ^a   Lee Soo, Jeoung ^a   Kim, Young Mi ^a  

^a Pusan National University   (South Korea)

Author keywords

5 Aminosalicyl L aspartic acid; 5 Aminosalicyl L glutamic acid; Colonspecific prodrug of 5 aminosalicylic acid; Inflammatory bowel disease

Indexed keywords

5 AMINOSALICYLASPARTIC ACID; 5 AMINOSALICYLGLUTAMIC ACID; AMINOSALICYLIC ACID DERIVATIVE; MESALAZINE; PRODRUG; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG BLOOD LEVEL; DRUG DISTRIBUTION; DRUG FECES LEVEL; DRUG SYNTHESIS; DRUG URINE LEVEL; IN VITRO STUDY; IN VIVO STUDY; LARGE INTESTINE; MALE; NONHUMAN; RAT;

EID: 0035155157     PISSN: 00223549     EISSN: None     Source Type: Journal    
DOI: 10.1002/jps.1126     Document Type: Article

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