Design, synthesis and antihistaminic (H1)activity of some condensed 2-(substituted)arylaminoethyl pyrimidin-4 (3H)-ones

Arzneimittel-Forschung/Drug Research

Volumn 51, Issue 3, 2001, Pages 221-231

  Shishoo, C J ^a   Shirsath, V S ^a   Rathod, I S ^a   Patil, M J ^a   Bhargava, S S ^a  

^a Gulbai Tekra   (India)

Author keywords

Antihistaminics; H1 antagonists; Pyrimidines, condensed, molecular modeling

Indexed keywords

4 AMINOTHIENOPYRIMIDINE DERIVATIVE; 4 OXOQUINAZOLINE DERIVATIVE; 4 OXOTHIENOPYRIMIDINE DERIVATIVE; ACETYLCHOLINE; AMINOETHYLPYRIMIDIN 4(3H) ONE DERIVATIVE; CETIRIZINE; HISTAMINE; HISTAMINE H1 RECEPTOR; HISTAMINE H1 RECEPTOR ANTAGONIST; TEMELASTINE; TERFENADINE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; ASPHYXIA; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DESIGN; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; GUINEA PIG; ILEUM CONTRACTION; IN VIVO STUDY; MALE; MOLECULAR MODEL; MOUSE; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION; SEDATION;

EID: 0035080118     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-0031-1300028     Document Type: Article

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