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Volumn 45, Issue 6, 2001, Pages 1682-1687

Pharmacokinetic-pharmacodynamic modeling of the electroencephalogram effect of imipenem in healthy rats

Author keywords

[No Author keywords available]

Indexed keywords

IMIPENEM;

EID: 0035006333     PISSN: 00664804     EISSN: None     Source Type: Journal    
DOI: 10.1128/AAC.45.6.1682-1687.2001     Document Type: Article
Times cited : (17)

References (41)
  • 1
    • 0021824648 scopus 로고
    • Review of adverse experiences and tolerability in the first 2,516 patients treated with imipenem/cilastatin
    • Calandra, G. B., K. R. Brown, L. C. Grad, V. I. Ahonkkai, C. Wang, and M. A. Aziz. 1985. Review of adverse experiences and tolerability in the first 2,516 patients treated with imipenem/cilastatin. Am. J. Med. 78(Suppl. 6A): 73-78.
    • (1985) Am. J. Med. , vol.78 , Issue.SUPPL. 6A , pp. 73-78
    • Calandra, G.B.1    Brown, K.R.2    Grad, L.C.3    Ahonkkai, V.I.4    Wang, C.5    Aziz, M.A.6
  • 2
    • 0023892181 scopus 로고
    • Factors predisposing to seizures in seriously ill infected patients receiving antibiotics: Experience with imipenem/cilastatin
    • Calandra, G. B., E. Lydick, J. Carrigan, L. Weiss, and H. Guess. 1988. Factors predisposing to seizures in seriously ill infected patients receiving antibiotics: experience with imipenem/cilastatin. Am. J. Med. 84:911-918.
    • (1988) Am. J. Med. , vol.84 , pp. 911-918
    • Calandra, G.B.1    Lydick, E.2    Carrigan, J.3    Weiss, L.4    Guess, H.5
  • 3
    • 0022971332 scopus 로고
    • The safety profile of imipenem/cilasatin: Worldwide clinical experience based on 3470 patients
    • Calandra, G. B., C. Wang, M. A. Aziz, and K. R. Brown. 1986. The safety profile of imipenem/cilasatin: worldwide clinical experience based on 3470 patients. J. Antimicrob. Chemother. 18(Suppl. E.):193-202.
    • (1986) J. Antimicrob. Chemother. , vol.18 , Issue.SUPPL. E , pp. 193-202
    • Calandra, G.B.1    Wang, C.2    Aziz, M.A.3    Brown, K.R.4
  • 4
    • 0025171043 scopus 로고
    • Determination of imipenem in human plasma, urine and tissue by high-performance liquid chromatography
    • Carlucci, G., L. Biordi, C. Vicentini, and M. Bologna. 1990. Determination of imipenem in human plasma, urine and tissue by high-performance liquid chromatography. J. Pharm. Biomed. Anal. 8:283-286.
    • (1990) J. Pharm. Biomed. Anal. , vol.8 , pp. 283-286
    • Carlucci, G.1    Biordi, L.2    Vicentini, C.3    Bologna, M.4
  • 5
    • 0025114459 scopus 로고
    • Central nervous system toxicity of quinolones: Human and animal findings
    • Christ, W. 1990. Central nervous system toxicity of quinolones: human and animal findings. J. Antimicrob. Chemother. 26(Suppl. B):219-225.
    • (1990) J. Antimicrob. Chemother. , vol.26 , Issue.SUPPL. B , pp. 219-225
    • Christ, W.1
  • 6
    • 0031936583 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic modeling of the electroencephalogram effect of synthetic opioids in the rat: Correlation with the interaction at the Mu-opioid receptor
    • Cox, E. H., T. Kerbusch, P. H. Van Der Graaf, and M. Danhof. 1998. Pharmacokinetic-pharmacodynamic modeling of the electroencephalogram effect of synthetic opioids in the rat: correlation with the interaction at the Mu-opioid receptor. J. Pharmacol. Exp. Ther. 284:1095-1103.
    • (1998) J. Pharmacol. Exp. Ther. , vol.284 , pp. 1095-1103
    • Cox, E.H.1    Kerbusch, T.2    Van Der Graaf, P.H.3    Danhof, M.4
  • 7
    • 0021276082 scopus 로고
    • Kinetics of drug action in disease states. 1. Effect of infusion rate on phenobarbital concentrations in serum, brain and cerebrospinal fluid of normal rats at onset of loss of righting reflex
    • Danhof, M., and G. Levy. 1984. Kinetics of drug action in disease states. 1. Effect of infusion rate on phenobarbital concentrations in serum, brain and cerebrospinal fluid of normal rats at onset of loss of righting reflex. J. Pharmacol. Exp. Ther. 229:44-50.
    • (1984) J. Pharmacol. Exp. Ther. , vol.229 , pp. 44-50
    • Danhof, M.1    Levy, G.2
  • 8
    • 0028965803 scopus 로고
    • Correlation between in vitro and in vivo models of proconvulsive activity with the carbapenem antibiotics, biapenem, imipenem/cilastatin and meropenem
    • Day, I. P., J. Goudie, K. Nishiki, and P. D. Williams. 1994. Correlation between in vitro and in vivo models of proconvulsive activity with the carbapenem antibiotics, biapenem, imipenem/cilastatin and meropenem. Toxicol. Lett. 76:239-243.
    • (1994) Toxicol. Lett. , vol.76 , pp. 239-243
    • Day, I.P.1    Goudie, J.2    Nishiki, K.3    Williams, P.D.4
  • 9
    • 0027769745 scopus 로고
    • Comparison of four basic models of indirect pharmacodynamic responses
    • Dayneka, N. L., V. Garg, and W. J. Jusko. 1993. Comparison of four basic models of indirect pharmacodynamic responses. J. Pharmacokinet. Biopharm. 21:457-478.
    • (1993) J. Pharmacokinet. Biopharm. , vol.21 , pp. 457-478
    • Dayneka, N.L.1    Garg, V.2    Jusko, W.J.3
  • 10
    • 0031885595 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic modeling of the anticonvulsant and electroencephalogram effects of phenytoin in rats
    • Della Paschoa, O. E., J. W. Mandema, R. A. Voskuyl, and M. Danhof. 1998. Pharmacokinetic-pharmacodynamic modeling of the anticonvulsant and electroencephalogram effects of phenytoin in rats. J. Pharmacol. Exp. Ther. 284:460-466.
    • (1998) J. Pharmacol. Exp. Ther. , vol.284 , pp. 460-466
    • Della Paschoa, O.E.1    Mandema, J.W.2    Voskuyl, R.A.3    Danhof, M.4
  • 11
    • 0033063077 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic contributions to the convulsant activity of fluoroquinolones in rats
    • Delon, A., S. Bouquet, F. Huguet, V. Brunet, P. Courtois, and W. Couet. 1999. Pharmacokinetic-pharmacodynamic contributions to the convulsant activity of fluoroquinolones in rats. Antimicrob. Agents Chemother. 43: 1511-1515.
    • (1999) Antimicrob. Agents Chemother. , vol.43 , pp. 1511-1515
    • Delon, A.1    Bouquet, S.2    Huguet, F.3    Brunet, V.4    Courtois, P.5    Couet, W.6
  • 12
    • 0031000142 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic contributions to the convulsant activity of pefloxacin and norfloxacin in rats
    • Delon, A., F. Huguet, P. Courtois, J. M. Vierfond, S. Bouquet, and W. Couet. 1997. Pharmacokinetic-pharmacodynamic contributions to the convulsant activity of pefloxacin and norfloxacin in rats. J. Pharmacol. Exp. Ther. 280: 983-987.
    • (1997) J. Pharmacol. Exp. Ther. , vol.280 , pp. 983-987
    • Delon, A.1    Huguet, F.2    Courtois, P.3    Vierfond, J.M.4    Bouquet, S.5    Couet, W.6
  • 13
    • 0033428350 scopus 로고    scopus 로고
    • Antagonistic interaction between the convulsant activities of pefloxacin and its main metabolite norfloxacin in rats
    • Delon, A., L. M. Levasseur, M. Giraudon, S. Bouquet, and W. Couet. 1999. Antagonistic interaction between the convulsant activities of pefloxacin and its main metabolite norfloxacin in rats. Pharm. Res. 16:1894-1897.
    • (1999) Pharm. Res. , vol.16 , pp. 1894-1897
    • Delon, A.1    Levasseur, L.M.2    Giraudon, M.3    Bouquet, S.4    Couet, W.5
  • 14
    • 0028216141 scopus 로고
    • Effects of some quinolones on imipenem induced-seizures in DBA/2 mice
    • De Sarro, A., D. Ammendola, and G. De Sarro. 1994. Effects of some quinolones on imipenem induced-seizures in DBA/2 mice. Gen. Pharmacol. 25:369-379.
    • (1994) Gen. Pharmacol. , vol.25 , pp. 369-379
    • De Sarro, A.1    Ammendola, D.2    De Sarro, G.3
  • 15
    • 0028817342 scopus 로고
    • Relationship between structure and convulsant properties of some β-lactam antibiotics following intracerebroventricular microinjection in rats
    • De Sarro, A., D. Ammendola, M. Zappala, S. Grasso, and G. B. De Sarro. 1995. Relationship between structure and convulsant properties of some β-lactam antibiotics following intracerebroventricular microinjection in rats. Antimicrob. Agents Chemother. 39:232-237.
    • (1995) Antimicrob. Agents Chemother. , vol.39 , pp. 232-237
    • De Sarro, A.1    Ammendola, D.2    Zappala, M.3    Grasso, S.4    De Sarro, G.B.5
  • 16
    • 0028954180 scopus 로고
    • Comparative convulsant potencies of two carbapenem derivatives in C57 and DBA/2 mice
    • De Sarro, A., C. Imperatore, P. Mastroeni, and G. De Sarro. 1995. Comparative convulsant potencies of two carbapenem derivatives in C57 and DBA/2 mice. J. Pharm. Pharmacol. 47:292-296.
    • (1995) J. Pharm. Pharmacol. , vol.47 , pp. 292-296
    • De Sarro, A.1    Imperatore, C.2    Mastroeni, P.3    De Sarro, G.4
  • 17
    • 0031039941 scopus 로고    scopus 로고
    • Effects of some excitatory amino acid antagonists and drugs enhancing γ-aminobutyric acid neurotransmission on pefloxacin-induced seizures in DBA/2 mice
    • De Sarro, G., B. F. Nava, G. Calapai, and A. De Sarro. 1997. Effects of some excitatory amino acid antagonists and drugs enhancing γ-aminobutyric acid neurotransmission on pefloxacin-induced seizures in DBA/2 mice. Antimicrob. Agents Chemother. 41:427-434.
    • (1997) Antimicrob. Agents Chemother. , vol.41 , pp. 427-434
    • De Sarro, G.1    Nava, B.F.2    Calapai, G.3    De Sarro, A.4
  • 18
    • 0022470510 scopus 로고
    • Imipenem-cilastatin. the promise of single agent antimicrobial therapy fulfilled?
    • Dudley, M. N. 1989. Imipenem-cilastatin. The promise of single agent antimicrobial therapy fulfilled? Clin. Pharm. 5:760.
    • (1989) Clin. Pharm. , vol.5 , pp. 760
    • Dudley, M.N.1
  • 20
    • 0034074059 scopus 로고    scopus 로고
    • Imipenem but not meropenem induces convulsions in DBA/2 mice, unrelated to cerebrospinal fluid concentrations
    • Dupuis, A., C. Pariat, P. Courtois, W. Couet, and S. Bouquet. 2000. Imipenem but not meropenem induces convulsions in DBA/2 mice, unrelated to cerebrospinal fluid concentrations. Fundam. Clin. Pharmacol. 14:163-165.
    • (2000) Fundam. Clin. Pharmacol. , vol.14 , pp. 163-165
    • Dupuis, A.1    Pariat, C.2    Courtois, P.3    Couet, W.4    Bouquet, S.5
  • 22
    • 0022642631 scopus 로고
    • Cerebrospinal fluid penetration of imipenem and cilastatin (Primaxin) in children with central nervous system infections
    • Jacobs, R. F., G. L. Kearns, A. L. Brown, and D. C. Longee. 1986. Cerebrospinal fluid penetration of imipenem and cilastatin (Primaxin) in children with central nervous system infections. Antimicrob. Agents Chemother. 29: 670-674.
    • (1986) Antimicrob. Agents Chemother. , vol.29 , pp. 670-674
    • Jacobs, R.F.1    Kearns, G.L.2    Brown, A.L.3    Longee, D.C.4
  • 23
    • 0027943266 scopus 로고
    • Physiologic indirect response models characterize diverse types of pharmacodynamic effects
    • Jusko, W. J., and H. C. Ko. 1994. Physiologic indirect response models characterize diverse types of pharmacodynamic effects. Clin. Pharmacol. Ther. 56:406-419.
    • (1994) Clin. Pharmacol. Ther. , vol.56 , pp. 406-419
    • Jusko, W.J.1    Ko, H.C.2
  • 24
    • 0025827837 scopus 로고
    • Seizure activity associated with imipenem use: Clinical case reports and review of the literature
    • Leo, R. J., and C. H. Ballow. 1991. Seizure activity associated with imipenem use: clinical case reports and review of the literature. DICP Ann, Pharmacother. 25:351-354.
    • (1991) DICP Ann, Pharmacother. , vol.25 , pp. 351-354
    • Leo, R.J.1    Ballow, C.H.2
  • 25
    • 0031817728 scopus 로고    scopus 로고
    • Development of a new quantitative approach for the isobolographic assessment of the convulsant interaction between pefloxacin and theophylline in rats
    • Levasseur, L. M., A. Delon, W. R. Greco, P. Faury, S. Bouquet, and W. Couet. 1998. Development of a new quantitative approach for the isobolographic assessment of the convulsant interaction between pefloxacin and theophylline in rats. Pharm. Res. 15:1069-1076.
    • (1998) Pharm. Res. , vol.15 , pp. 1069-1076
    • Levasseur, L.M.1    Delon, A.2    Greco, W.R.3    Faury, P.4    Bouquet, S.5    Couet, W.6
  • 26
    • 0026058369 scopus 로고
    • Pharmacokinetic-pharmacodynamic modelling of the EEG effects of midazolam in individual rats: Influence of rate and route of administration
    • Mandema, J. W., E. Tukker, and M. Danhof. 1991. Pharmacokinetic-pharmacodynamic modelling of the EEG effects of midazolam in individual rats: influence of rate and route of administration. Br. J. Pharmacol. 102:663-668.
    • (1991) Br. J. Pharmacol. , vol.102 , pp. 663-668
    • Mandema, J.W.1    Tukker, E.2    Danhof, M.3
  • 27
    • 0034002147 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic modelling of the convulsant interaction between norfloxacin and biphenyl acetic acid in rats
    • Marchand, S., C. Pariat, S. Bouquet, P. Courtois, and W. Couet. 2000. Pharmacokinetic-pharmacodynamic modelling of the convulsant interaction between norfloxacin and biphenyl acetic acid in rats. Brit. J. Pharmacol. 129:1609-1616.
    • (2000) Brit. J. Pharmacol. , vol.129 , pp. 1609-1616
    • Marchand, S.1    Pariat, C.2    Bouquet, S.3    Courtois, P.4    Couet, W.5
  • 28
    • 0022408794 scopus 로고
    • Penetration of imipenem and cilastatin into cerebrospinal fluid of patients with bacterial meningitis
    • Modai, J., D. Vittecoq, J. M. Decazes, and A. Meulemans. 1985. Penetration of imipenem and cilastatin into cerebrospinal fluid of patients with bacterial meningitis. J. Antimicrob. Chemother. 16:751-755.
    • (1985) J. Antimicrob. Chemother. , vol.16 , pp. 751-755
    • Modai, J.1    Vittecoq, D.2    Decazes, J.M.3    Meulemans, A.4
  • 29
    • 0029823378 scopus 로고    scopus 로고
    • Neurotoxicity of carbapenem antibacterials
    • Norrby, R. S. 1996. Neurotoxicity of carbapenem antibacterials. Drug Saf. 15:87-90.
    • (1996) Drug Saf. , vol.15 , pp. 87-90
    • Norrby, R.S.1
  • 30
    • 0024415132 scopus 로고
    • Meropenem: Evidence of lack of proconvulsive tendency in mice
    • Patel, J. B., and R. E. Giles. 1989. Meropenem: evidence of lack of proconvulsive tendency in mice. J. Antimicrob. Chemother. 24(Suppl. A):307-309.
    • (1989) J. Antimicrob. Chemother. , vol.24 , Issue.SUPPL. A , pp. 307-309
    • Patel, J.B.1    Giles, R.E.2
  • 31
    • 0021921241 scopus 로고
    • Kinetics of drug action in disease states. XIV. Effect of infusion rate on pentylenetetrazol concentrations in serum, brain and cerebrospinal fluid of rats at onset of convulsions
    • Ramzan, I. M., and G. Levy. 1985. Kinetics of drug action in disease states. XIV. Effect of infusion rate on pentylenetetrazol concentrations in serum, brain and cerebrospinal fluid of rats at onset of convulsions. J. Pharmacol. Exp. Ther. 234:624-628.
    • (1985) J. Pharmacol. Exp. Ther. , vol.234 , pp. 624-628
    • Ramzan, I.M.1    Levy, G.2
  • 32
    • 0022491959 scopus 로고
    • Kinetics of drug action in disease states. XVI. Pharmacodynamics of theophylline induced seizures in rats
    • Ramzan, I. M., and G. Levy. 1986. Kinetics of drug action in disease states. XVI. Pharmacodynamics of theophylline induced seizures in rats. J. Pharmacol. Exp. Ther. 236:708-713.
    • (1986) J. Pharmacol. Exp. Ther. , vol.236 , pp. 708-713
    • Ramzan, I.M.1    Levy, G.2
  • 33
    • 0025828473 scopus 로고
    • Neurotoxicity of β-lactam: Predisposing factors and pathogenesis
    • Schliamser, S. E., O. Cars, and S. R. Norrby. 1991. Neurotoxicity of β-lactam: predisposing factors and pathogenesis. J. Antimicrob. Chemother. 27: 405-425.
    • (1991) J. Antimicrob. Chemother. , vol.27 , pp. 405-425
    • Schliamser, S.E.1    Cars, O.2    Norrby, S.R.3
  • 34
    • 0030429755 scopus 로고    scopus 로고
    • Characterization of four basic models of indirect pharmacodynamic responses
    • Sharma, A., and W. J. Jusko. 1996. Characterization of four basic models of indirect pharmacodynamic responses. J. Pharmacokinet. Biopharm. 24:611-635.
    • (1996) J. Pharmacokinet. Biopharm. , vol.24 , pp. 611-635
    • Sharma, A.1    Jusko, W.J.2
  • 35
    • 0018394195 scopus 로고
    • Simultaneous modelling of pharmacokinetics and pharmacodynamics: Application to d-tubocurarine
    • Sheiner, L. B., D. R. Stanski, S. Vozeh, R. D. Miller, and J. Ham. 1979. Simultaneous modelling of pharmacokinetics and pharmacodynamics: application to d-tubocurarine. Clin. Pharmacol. Ther. 25:358-371.
    • (1979) Clin. Pharmacol. Ther. , vol.25 , pp. 358-371
    • Sheiner, L.B.1    Stanski, D.R.2    Vozeh, S.3    Miller, R.D.4    Ham, J.5
  • 36
    • 0029046103 scopus 로고
    • Structural features resulting in convulsive activity of carbapenem compounds: Effect of C-2 side chain
    • Sunagawa, M., H. Matsumura, Y. Sumita, and H. Nouda. 1995. Structural features resulting in convulsive activity of carbapenem compounds: effect of C-2 side chain. J. Antibiot. 48:408-416.
    • (1995) J. Antibiot. , vol.48 , pp. 408-416
    • Sunagawa, M.1    Matsumura, H.2    Sumita, Y.3    Nouda, H.4
  • 37
    • 0023279701 scopus 로고
    • Seizure-like activity associated with imipenem-cilastatin
    • Tse, C. S. T., F. H. Vera, and D. V. Desai. 1987. Seizure-like activity associated with imipenem-cilastatin. Drug Intell. Clin. Pharm. 21:659-660.
    • (1987) Drug Intell. Clin. Pharm. , vol.21 , pp. 659-660
    • Tse, C.S.T.1    Vera, F.H.2    Desai, D.V.3
  • 38
    • 0031881728 scopus 로고    scopus 로고
    • The time of maximum effect for model selection in pharmacokinetic-pharmacodynamic analysis applied to frusemide
    • Wakelkamp, M., G. Alvan, and G. Paintaud. 1998. The time of maximum effect for model selection in pharmacokinetic-pharmacodynamic analysis applied to frusemide. Br. J. Clin. Pharmacol. 45:63-70.
    • (1998) Br. J. Clin. Pharmacol. , vol.45 , pp. 63-70
    • Wakelkamp, M.1    Alvan, G.2    Paintaud, G.3
  • 39
    • 0030747113 scopus 로고    scopus 로고
    • Antibiotic-induced convulsions
    • Wallace, K. L. 1997. Antibiotic-induced convulsions. Crit. Care Clin. 13:741-762.
    • (1997) Crit. Care Clin. , vol.13 , pp. 741-762
    • Wallace, K.L.1
  • 40
    • 0023947514 scopus 로고
    • Animal model for evaluating the convulsive liability of β-lactam antibiotics
    • Williams, P. D., D. B. Bennett, and C. R. Comereski. 1988. Animal model for evaluating the convulsive liability of β-lactam antibiotics. Antimicrob. Agents Chemother. 32:758-760.
    • (1988) Antimicrob. Agents Chemother. , vol.32 , pp. 758-760
    • Williams, P.D.1    Bennett, D.B.2    Comereski, C.R.3


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