Key structural features of prostaglandin E2 and prostanoid analogs involved in binding and activation of the human EP1 prostanoid receptor

Molecular Pharmacology

Volumn 59, Issue 6, 2001, Pages 1446-1456

  Ungrin, M D ^a   Carriere M C ^a   Denis, D ^a   Lamontagne, S ^a   Sawyer, N ^a   Stocco, R ^a   Tremblay, N ^a   Metters, K M ^a   Abramovitz, M ^a  

^a MERCK FROSST CENTRE FOR THERAPEUTIC RESEARCH   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

9 DEOXY 9 METHYLENEPROSTAGLANDIN E2; CARBOXYLIC ACID; HYDROXYL GROUP; PROSTAGLANDIN E2; PROSTANOID; PROSTANOID DERIVATIVE; PROSTANOID RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CELL LINE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG BINDING; DRUG DETERMINATION; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG TOLERABILITY; EMBRYO; HUMAN; HUMAN CELL; KIDNEY CELL; PRIORITY JOURNAL; PROTEIN EXPRESSION; STRUCTURE ACTIVITY RELATION;

EID: 0034981519     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.59.6.1446     Document Type: Article

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