SCOPUS 정보 검색 플랫폼

Volumn 28, Issue 6, 2001, Pages 639-643

In vivo evaluation of 4-[123I]iodo-N-(2-[4-(6-trifluoromethyl-2-pyridinyl)-1- piperazinyl]ethyl)benzamide, a potential SPECT radioligand for the 5-HT1A receptor

(8) Vandecapelle, M a De Vos, F a Vermeirsch, H a De Ley, G a Audenaert, K a Leysen, D a Dierckx, R A a Slegers, G a

a GHENT UNIVERSITY (Belgium)

Author keywords

5 HT1A agonist; 123I labeling; Biodistribution study; Blocking experiments

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 4 FLUORO N [2 [4 (6 TRIFLUOROMETHYL 2 PYRIDINYL) 1 PIPERAZINYL]ETHYL]BENZAMIDE; 4 IODO N [2 [4 (6 TRIFLUOROMETHYL 2 PYRIDINYL) 1 PIPERAZINYL]ETHYL]BENZAMIDE; BENZAMIDE DERIVATIVE; IODINE 123; KETANSERIN; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; RADIOLIGAND; SEROTONIN 1A AGONIST; SEROTONIN 1A RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN REGION; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG DISTRIBUTION; IN VIVO STUDY; ISOTOPE LABELING; LIPOPHILICITY; NONHUMAN; RADIOACTIVITY; RAT; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY; SYNTHESIS; TISSUE DISTRIBUTION;

8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN; ANIMALS; BENZAMIDES; BRAIN; KETANSERIN; MALE; PIPERAZINES; PYRIDINES; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED, SINGLE-PHOTON;

EID: 0034888413 PISSN: 09698051 EISSN: None Source Type: Journal
DOI: 10.1016/S0969-8051(01)00223-2 Document Type: Article

Times cited : (12)

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