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Quantitative Structure-Activity Relationships

Volumn 20, Issue 2, 2001, Pages 130-138

Human P-glycoprotein pseudoreceptor modeling: 3D-QSAR study on thioxanthene type multidrug resistance modulators

(2) Pajeva, Ilza K a Wiese, Michael b

a BULGARIAN ACADEMY OF SCIENCES (Bulgaria)

b UNIVERSITY OF BONN (Germany)

Author keywords

3D QSAR; MDR, P glycoprotein; Pseudoreceptor modeling

Indexed keywords

ACTIVATION ANALYSIS; GLYCOPROTEINS; HYDROPHOBICITY; INSECTICIDES;

3D-QSAR; DOMAIN MODEL; EXTENDED MODEL; HYDROPHOBICS; MULTIDRUG RESISTANCE; MULTIDRUG RESISTANCE, P-GLYCOPROTEIN; P-GLYCOPROTEIN; PSEUDORECEPTOR MODEL; SINGLE DOMAINS; THIOXANTHENE;

LIGANDS;

GLYCOPROTEIN P; PHENOTHIAZINE DERIVATIVE; THIOXANTHENE DERIVATIVE;

ARTICLE; DRUG STRUCTURE; GENE MUTATION; HUMAN; HYDROGEN BOND; HYDROPHOBICITY; MODEL; MULTIDRUG RESISTANCE; PRIORITY JOURNAL; QUANTITATIVE STRUCTURE ACTIVITY RELATION;

EID: 0034868283 PISSN: 09318771 EISSN: None Source Type: Journal
DOI: 10.1002/1521-3838(200107)20:2<130::AID-QSAR130>3.0.CO;2-6 Document Type: Article

Times cited : (15)

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