-
1
-
-
0028149954
-
Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1
-
Borden L.A., Murali Dhar T.G., Smith K.E., Weinshank R.L., Branchek T.A., Gluchowski C. Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1. Eur. J. Pharmacol. 269:1994;219-224.
-
(1994)
Eur. J. Pharmacol.
, vol.269
, pp. 219-224
-
-
Borden, L.A.1
Murali Dhar, T.G.2
Smith, K.E.3
Weinshank, R.L.4
Branchek, T.A.5
Gluchowski, C.6
-
2
-
-
0025068791
-
(R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acid binds with high affinity to the brain gamma-aminobutyric acid uptake carrier
-
Braestrup C., Nielsen E.B., Sonnewald U., Knutsen L.J., Andersen K.E., Jansen J.A., Frederiksen K., Andersen P.H., Mortensen A., Suzdak P.D. (R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acid binds with high affinity to the brain gamma-aminobutyric acid uptake carrier. J. Neurochem. 54:1990;639-647.
-
(1990)
J. Neurochem.
, vol.54
, pp. 639-647
-
-
Braestrup, C.1
Nielsen, E.B.2
Sonnewald, U.3
Knutsen, L.J.4
Andersen, K.E.5
Jansen, J.A.6
Frederiksen, K.7
Andersen, P.H.8
Mortensen, A.9
Suzdak, P.D.10
-
3
-
-
0032894933
-
Effects of baclofen on maintenance and reinstatement of intravenous cocaine self-administration in rats
-
Campbell U.C., Lac S.T., Carroll M.E. Effects of baclofen on maintenance and reinstatement of intravenous cocaine self-administration in rats. Psychopharmacology. 143:1999;209-214.
-
(1999)
Psychopharmacology
, vol.143
, pp. 209-214
-
-
Campbell, U.C.1
Lac, S.T.2
Carroll, M.E.3
-
4
-
-
0025782810
-
Inhibition of famma-aminobutyrate and glycine uptake into synaptic vesicles
-
Christensen H., Fykse E.M., Fonnum F. Inhibition of famma-aminobutyrate and glycine uptake into synaptic vesicles. Eur. J. Pharmacol. 207:1991;73-79.
-
(1991)
Eur. J. Pharmacol.
, vol.207
, pp. 73-79
-
-
Christensen, H.1
Fykse, E.M.2
Fonnum, F.3
-
5
-
-
0029884812
-
Benzodiazepines on trial: A research stragegy for their rehabilitation
-
Costa E., Guidotti A. Benzodiazepines on trial: a research stragegy for their rehabilitation. TIPS. 17:1996;192-200.
-
(1996)
TIPS
, vol.17
, pp. 192-200
-
-
Costa, E.1
Guidotti, A.2
-
6
-
-
0024437218
-
Long term evaluation of vigabatrin (gamma vinyl-GABA) in epilepsy
-
Dam M. Long term evaluation of vigabatrin (gamma vinyl-GABA) in epilepsy. Epilepsia. 30:1989;S26-S30.
-
(1989)
Epilepsia
, vol.30
, pp. 26-S30
-
-
Dam, M.1
-
7
-
-
0026707806
-
GABAergic inhibition of endogenous dopamine release measured in vivo with 11C-raclopride and positron emission tomography
-
Dewey S.L., Smith G.S., Logan J., Brodie J.D., Yu D.W., Ferrieri R.A., King P.T., MacGregor R.R., Martin T.P., Wolf A.P. GABAergic inhibition of endogenous dopamine release measured in vivo with 11C-raclopride and positron emission tomography. J. Neurosci. 12:1992;3773-3780.
-
(1992)
J. Neurosci.
, vol.12
, pp. 3773-3780
-
-
Dewey, S.L.1
Smith, G.S.2
Logan, J.3
Brodie, J.D.4
Yu, D.W.5
Ferrieri, R.A.6
King, P.T.7
MacGregor, R.R.8
Martin, T.P.9
Wolf, A.P.10
-
8
-
-
0030975733
-
GABAergic attenuation of cocaine-induced dopamine release and locomotor activity
-
Dewey S.L., Chaurasia C.S., Chen C.E., Volkow N.D., Clarkson F.A., Porter S.P., Straughter-Moore R.M., Alexoff D.L., Tedeschi D., Russo N.B., Fowler J.S., Brodie J.D. GABAergic attenuation of cocaine-induced dopamine release and locomotor activity. Synapse. 25:1997;393-398.
-
(1997)
Synapse
, vol.25
, pp. 393-398
-
-
Dewey, S.L.1
Chaurasia, C.S.2
Chen, C.E.3
Volkow, N.D.4
Clarkson, F.A.5
Porter, S.P.6
Straughter-Moore, R.M.7
Alexoff, D.L.8
Tedeschi, D.9
Russo, N.B.10
Fowler, J.S.11
Brodie, J.D.12
-
9
-
-
7344221467
-
A novel strategy for the treatment of cocaine addiction
-
Dewey S.L., Morgan A.E., Ashby C.R.J., Horan B., Kushner S.A., Logan J., Volkow N.D., Fowler J.S., Gardner E.L., Brodie J.D. A novel strategy for the treatment of cocaine addiction. Synapse. 30:1998;119-129.
-
(1998)
Synapse
, vol.30
, pp. 119-129
-
-
Dewey, S.L.1
Morgan, A.E.2
Ashby, C.R.J.3
Horan, B.4
Kushner, S.A.5
Logan, J.6
Volkow, N.D.7
Fowler, J.S.8
Gardner, E.L.9
Brodie, J.D.10
-
10
-
-
0032908565
-
A pharmacologic strategy for the treatment of nicotine addiction
-
Dewey S.L., Brodie J.D., Gerasimov M., Horan B., Gardner E.L., Ashby C.R.J. A pharmacologic strategy for the treatment of nicotine addiction. Synapse. 31:1999;76-86.
-
(1999)
Synapse
, vol.31
, pp. 76-86
-
-
Dewey, S.L.1
Brodie, J.D.2
Gerasimov, M.3
Horan, B.4
Gardner, E.L.5
Ashby, C.R.J.6
-
11
-
-
0027329888
-
GABA(B) receptor activation alters the firing pattern of dopamine neurons in the rat substantia nigra
-
Engberg G., Klingpetersen T., Nissbrandt H. GABA(B) receptor activation alters the firing pattern of dopamine neurons in the rat substantia nigra. Synapse. 15:1993;229-238.
-
(1993)
Synapse
, vol.15
, pp. 229-238
-
-
Engberg, G.1
Klingpetersen, T.2
Nissbrandt, H.3
-
12
-
-
0026709603
-
The gamma-aminobutyric acid (GABA) uptake inhibitor, tiagabine, increases extracellular brain levels of GABA in awake rats
-
Fink-Jensen A., Suzdak P.D., Swedberg M.D., Judge M.E., Hansen L., Nielsen P.G. The gamma-aminobutyric acid (GABA) uptake inhibitor, tiagabine, increases extracellular brain levels of GABA in awake rats. Eur. J. Pharmacol. 220:1992;197-201.
-
(1992)
Eur. J. Pharmacol.
, vol.220
, pp. 197-201
-
-
Fink-Jensen, A.1
Suzdak, P.D.2
Swedberg, M.D.3
Judge, M.E.4
Hansen, L.5
Nielsen, P.G.6
-
13
-
-
0026580109
-
Benzodiazepine-induced decreases in extracellular concentrations of dopamine in the nucleus accumbens after acute and repeated administration
-
Finlay J.M., Damsma G., Fibiger H.C. Benzodiazepine-induced decreases in extracellular concentrations of dopamine in the nucleus accumbens after acute and repeated administration. Psycopharmacology. 106:1992;202-208.
-
(1992)
Psycopharmacology
, vol.106
, pp. 202-208
-
-
Finlay, J.M.1
Damsma, G.2
Fibiger, H.C.3
-
14
-
-
0033214654
-
Gamma-vinyl GABA inhibits methamphetamine, heroin, or ethanol-induced increases in nucleus accumbens dopamine
-
Gerasimov M.R., Ashby C.R., Gardner E.L., Mills M.J., Brodie J.D., Dewey S.L. Gamma-vinyl GABA inhibits methamphetamine, heroin, or ethanol-induced increases in nucleus accumbens dopamine. Synapse. 34:1999;11-19.
-
(1999)
Synapse
, vol.34
, pp. 11-19
-
-
Gerasimov, M.R.1
Ashby, C.R.2
Gardner, E.L.3
Mills, M.J.4
Brodie, J.D.5
Dewey, S.L.6
-
15
-
-
0029916715
-
Effect of nucleus accumbens dopamine depletion on motivational aspects involved in initiation of cocaine and heroin self-administration in rats
-
Gerrits M.A., Van Ree J.M. Effect of nucleus accumbens dopamine depletion on motivational aspects involved in initiation of cocaine and heroin self-administration in rats. Brain Res. 713:1996;114-124.
-
(1996)
Brain Res.
, vol.713
, pp. 114-124
-
-
Gerrits, M.A.1
Van Ree, J.M.2
-
16
-
-
0032453937
-
A receptor modulator, inhibits the effects of cocaine on locomotor activity and extracellular dopamine in the nucleus accumbens shell without tolerance liability
-
A receptor modulator, inhibits the effects of cocaine on locomotor activity and extracellular dopamine in the nucleus accumbens shell without tolerance liability. J. Pharmacol. Exp. Ther. 287:1998;58-66.
-
(1998)
J. Pharmacol. Exp. Ther.
, vol.287
, pp. 58-66
-
-
Giorgetti, M.1
Javaid, J.I.2
Davis, J.M.3
Costa, E.4
Guidotti, A.5
Appel, S.B.6
Brodie, M.S.7
-
17
-
-
0031817159
-
GABAergic modulation of ventral pallidal dopamine release studied by in vivo microdialysis in the freely moving rat
-
Gong W., Neill D.B., Justice J.B.J. GABAergic modulation of ventral pallidal dopamine release studied by in vivo microdialysis in the freely moving rat. Synapse. 29:1998;406-412.
-
(1998)
Synapse
, vol.29
, pp. 406-412
-
-
Gong, W.1
Neill, D.B.2
Justice, J.B.J.3
-
18
-
-
0027050085
-
Acute effects of gamma-vinyl GABA on the GABAergic system in rats as studied by microdialysis
-
Jolkkonen J., Mazurkiewicz M., Lahtinen H., Riekkinen P. Acute effects of gamma-vinyl GABA on the GABAergic system in rats as studied by microdialysis. Eur. J. Pharmacol. 229:1992;269-272.
-
(1992)
Eur. J. Pharmacol.
, vol.229
, pp. 269-272
-
-
Jolkkonen, J.1
Mazurkiewicz, M.2
Lahtinen, H.3
Riekkinen, P.4
-
19
-
-
0017553966
-
Gamma-vinyl GABA (4-amino-hex-5-enoic acid), a new selective irreversible inhibitor of GABA-T: Effects on brain GABA metabolism in mice
-
Jung M.J., Lippert B., Metcalf B.W., Böhlen P., Schechter P.J. Gamma-vinyl GABA (4-amino-hex-5-enoic acid), a new selective irreversible inhibitor of GABA-T: effects on brain GABA metabolism in mice. J. Neurochem. 29:1977;797-802.
-
(1977)
J. Neurochem.
, vol.29
, pp. 797-802
-
-
Jung, M.J.1
Lippert, B.2
Metcalf, B.W.3
Böhlen, P.4
Schechter, P.J.5
-
20
-
-
0025346635
-
Modulation of A10 dopamine neurons by gamma-aminobutyric acid agonists
-
Kalivas P.W., Duffy P., Eberhardt H. Modulation of A10 dopamine neurons by gamma-aminobutyric acid agonists. J. Pharmacol. Exp. Ther. 253:1990;858-866.
-
(1990)
J. Pharmacol. Exp. Ther.
, vol.253
, pp. 858-866
-
-
Kalivas, P.W.1
Duffy, P.2
Eberhardt, H.3
-
21
-
-
0032241893
-
Tiagabine: A new therapeutic option for people with intellectual disability and partial epilepsy
-
Kälviäinen R. Tiagabine: a new therapeutic option for people with intellectual disability and partial epilepsy. J. Intellect. Disabil. Res. 42(Suppl. 1):1998;63-67.
-
(1998)
J. Intellect. Disabil. Res.
, vol.42
, pp. 63-67
-
-
Kälviäinen, R.1
-
22
-
-
0016837251
-
Inhibition of GABA uptake in rat brain slices by nipecotic acid, various isoxazoles and related compounds
-
Krogsgaard-Larsen P., Johnston G.A. Inhibition of GABA uptake in rat brain slices by nipecotic acid, various isoxazoles and related compounds. J. Neurochem. 25:1975;797-802.
-
(1975)
J. Neurochem.
, vol.25
, pp. 797-802
-
-
Krogsgaard-Larsen, P.1
Johnston, G.A.2
-
23
-
-
0025855256
-
The dopamine hypothesis of the reinforcing properties of cocaine
-
Kuhar M.J., Ritz M.C., Boja J.W. The dopamine hypothesis of the reinforcing properties of cocaine. TIPS. 14:1991;299-302.
-
(1991)
TIPS
, vol.14
, pp. 299-302
-
-
Kuhar, M.J.1
Ritz, M.C.2
Boja, J.W.3
-
24
-
-
0032765110
-
The irreversible gamma-aminobutyric acid (GABA) transaminase inhibitor gamma-vinyl GABA blocks cocaine self administration in rats
-
Kushner S.A., Dewey S.L., Kornetsky C. The irreversible gamma-aminobutyric acid (GABA) transaminase inhibitor gamma-vinyl GABA blocks cocaine self administration in rats. J. Pharmacol. Exp. Ther. 290:1999;797-802.
-
(1999)
J. Pharmacol. Exp. Ther.
, vol.290
, pp. 797-802
-
-
Kushner, S.A.1
Dewey, S.L.2
Kornetsky, C.3
-
25
-
-
0032904836
-
The effects of diazepam and zolpidem on cocaine- And amphetamine-induced place preference
-
Meririnne E., Kankaanpää A., Lillsunde P., Seppälä T. The effects of diazepam and zolpidem on cocaine- and amphetamine-induced place preference. Pharmacol. Biochem. Behav. 62:1999;159-164.
-
(1999)
Pharmacol. Biochem. Behav.
, vol.62
, pp. 159-164
-
-
Meririnne, E.1
Kankaanpää, A.2
Lillsunde, P.3
Seppälä, T.4
-
26
-
-
9844253326
-
Effects of pharmacologic increases in brain GABA levels on cocaine-induced changes in extracellular dopamine
-
Morgan A.E., Dewey S.L. Effects of pharmacologic increases in brain GABA levels on cocaine-induced changes in extracellular dopamine. Synapse. 28:1998;60-65.
-
(1998)
Synapse
, vol.28
, pp. 60-65
-
-
Morgan, A.E.1
Dewey, S.L.2
-
27
-
-
0030797532
-
Direct approach for attenuating cocaine's effects on extracellular dopamine: Targeting the dopamine transporter
-
Morgan A.E., Porter S.P., Clarkson F.A., Volkow N.D., Fowler J.S., Dewey S.L. Direct approach for attenuating cocaine's effects on extracellular dopamine: targeting the dopamine transporter. Synapse. 26:1997;423-427.
-
(1997)
Synapse
, vol.26
, pp. 423-427
-
-
Morgan, A.E.1
Porter, S.P.2
Clarkson, F.A.3
Volkow, N.D.4
Fowler, J.S.5
Dewey, S.L.6
-
28
-
-
0025805321
-
Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor
-
Nielsen E.B., Suzdak P.D., Andersen K.E., Knutsen L.J., Sonnewald U., Braestrup C. Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor. Eur. J. Pharmacol. 196:1991;257-266.
-
(1991)
Eur. J. Pharmacol.
, vol.196
, pp. 257-266
-
-
Nielsen, E.B.1
Suzdak, P.D.2
Andersen, K.E.3
Knutsen, L.J.4
Sonnewald, U.5
Braestrup, C.6
-
29
-
-
0027484607
-
Serotonin and dopamine sensitization in the nucleus accumbens, ventral tegmental area, and dorsal raphe nucleus following repeated cocaine administration
-
Parsons L.H., Justice J.B.J. Serotonin and dopamine sensitization in the nucleus accumbens, ventral tegmental area, and dorsal raphe nucleus following repeated cocaine administration. J. Neurochem. 61:1993;1611-1619.
-
(1993)
J. Neurochem.
, vol.61
, pp. 1611-1619
-
-
Parsons, L.H.1
Justice, J.B.J.2
-
30
-
-
0029953127
-
Human brain GABA levels rise after initiation of vigabatrin therapy but fail to rise further with increasing dose
-
Petroff O.A., Rothman D.L., Behar K.L., Mattson R.H. Human brain GABA levels rise after initiation of vigabatrin therapy but fail to rise further with increasing dose. Neurology. 46:1996;1459-1463.
-
(1996)
Neurology
, vol.46
, pp. 1459-1463
-
-
Petroff, O.A.1
Rothman, D.L.2
Behar, K.L.3
Mattson, R.H.4
-
31
-
-
0026011576
-
Effect of dose on cocaine self-administration behavior and dopamine levels in the nucleus accumbens
-
Pettit H.O., Justice J.B.J. Effect of dose on cocaine self-administration behavior and dopamine levels in the nucleus accumbens. Brain Res. 539:1991;94-102.
-
(1991)
Brain Res.
, vol.539
, pp. 94-102
-
-
Pettit, H.O.1
Justice, J.B.J.2
-
32
-
-
0025122568
-
Extracellular concentrations of cocaine and dopamine are enhanced during chronic cocaine administration
-
Pettit H.O., Pan H.T., Parsons L.H., Justice J.B.J. Extracellular concentrations of cocaine and dopamine are enhanced during chronic cocaine administration. J. Neurochem. 55:1990;798-804.
-
(1990)
J. Neurochem.
, vol.55
, pp. 798-804
-
-
Pettit, H.O.1
Pan, H.T.2
Parsons, L.H.3
Justice, J.B.J.4
-
33
-
-
84992614598
-
Inhibition and substrate activity of conformationally rigid vigabatrin analogues with gamma-aminobutyric acid aminotransferase
-
(in press)
-
Qui J., Pingstehaus J.M., Silverman R. Inhibition and substrate activity of conformationally rigid vigabatrin analogues with gamma-aminobutyric acid aminotransferase. J. Med. Chem. 2000;. (in press).
-
(2000)
J. Med. Chem.
-
-
Qui, J.1
Pingstehaus, J.M.2
Silverman, R.3
-
36
-
-
0020034196
-
Gamma-aminobutyric acid (GABA) receptor stimulation. III. Effect of progabide (SL 76002) on norepinephrine, dopamine and 5-hydroxytryptamine turnover in rat brain areas
-
Scatton B., Zivkovic B., Dedek J., Lloyd K.G., Constantinidis J., Tissot R., Bartholini G. Gamma-aminobutyric acid (GABA) receptor stimulation. III. Effect of progabide (SL 76002) on norepinephrine, dopamine and 5-hydroxytryptamine turnover in rat brain areas. J. Pharmacol. Exp. Ther. 220:1982;678-688.
-
(1982)
J. Pharmacol. Exp. Ther.
, vol.220
, pp. 678-688
-
-
Scatton, B.1
Zivkovic, B.2
Dedek, J.3
Lloyd, K.G.4
Constantinidis, J.5
Tissot, R.6
Bartholini, G.7
-
37
-
-
0026538586
-
Repeated cocaine administration induces behavioral sensitization and corresponding decreased extracellular dopamine responses in caudate and accumbens
-
Segal D.S., Kuczenski R. Repeated cocaine administration induces behavioral sensitization and corresponding decreased extracellular dopamine responses in caudate and accumbens. Brain Res. 577:1992;351-355.
-
(1992)
Brain Res.
, vol.577
, pp. 351-355
-
-
Segal, D.S.1
Kuczenski, R.2
-
38
-
-
0027753878
-
Lipophilic GABA uptake inhibitors: Biochemistry, pharmacology and therapeutic potential
-
Suzdak P.D. Lipophilic GABA uptake inhibitors: Biochemistry, pharmacology and therapeutic potential. Drugs Future. 18:1993;1129-1136.
-
(1993)
Drugs Future
, vol.18
, pp. 1129-1136
-
-
Suzdak, P.D.1
-
39
-
-
0026539825
-
NNC-711, a novel potent and selective gamma-aminobutyric acid uptake inhibitor: Pharmacological characterization
-
Suzdak P.D., Frederiksen K., Andersen K.E., Sørensen P.O., Knutsen L.J., Nielsen E.B. NNC-711, a novel potent and selective gamma-aminobutyric acid uptake inhibitor: pharmacological characterization. Eur. J. Pharmacol. 224:1992;189-198.
-
(1992)
Eur. J. Pharmacol.
, vol.224
, pp. 189-198
-
-
Suzdak, P.D.1
Frederiksen, K.2
Andersen, K.E.3
Sørensen, P.O.4
Knutsen, L.J.5
Nielsen, E.B.6
-
40
-
-
0030858106
-
Drug dependence study on vigabatrin in rhesus monkeys and rats
-
Takada K., Yanagita T. Drug dependence study on vigabatrin in rhesus monkeys and rats. Arzneim.-Forsch./Drug Res. 47:1997;1087-1092.
-
(1997)
Arzneim.-Forsch./Drug Res.
, vol.47
, pp. 1087-1092
-
-
Takada, K.1
Yanagita, T.2
-
41
-
-
0032490594
-
A receptors-an in vivo electrochemical study
-
A receptors-an in vivo electrochemical study. Brain Res. 798:1998;156-165.
-
(1998)
Brain Res.
, vol.798
, pp. 156-165
-
-
Xi, Z.X.1
Stein, E.A.2
|