Assessment of potential mutagenic activities of a novel benzothiazole MAO-A inhibitor E2011 using Salmonella typhimurium YG1029

Mutation Research - Genetic Toxicology and Environmental Mutagenesis

Volumn 472, Issue 1-2, 2000, Pages 163-169

  Sato, Gen ^a   Asakura, Shoji ^a   Hakura, Atsushi ^a   Tsutsui Hiyoshi, Yoshie ^a   Kobayashi, Naoki ^a   Tsukidate, Kazuo ^a  

^a EISAI CO LTD   (Japan)

Author keywords

Acetyltransferase; Aromatic amine; Benzothiazole; Decarbonation; E2011; Salmonella typhimurium

Indexed keywords

3 [2 (3 CYANO 1 HYDROXYPROPYL) 6 BENZOTHIAZOLYL] 5 METHOXYMETHYL 2 OXAZOLIDINONE; 6 AMINOBENZOTHIAZOLE; ACYLTRANSFERASE; AROMATIC AMINE; BENZOTHIAZOLE DERIVATIVE; ER 174237 00; ER 174238 00; MONOAMINE OXIDASE A INHIBITOR; MUTAGENIC AGENT; S 9; TERTIARY AMINE; UNCLASSIFIED DRUG;

AMES TEST; ARTICLE; CONTROLLED STUDY; DRUG STRUCTURE; LIVER TOXICITY; MUTAGENICITY; NONHUMAN; PRIORITY JOURNAL; SALMONELLA TYPHIMURIUM; STRAIN DIFFERENCE; STRUCTURE ACTIVITY RELATION;

ACETYLTRANSFERASES; ANIMALS; BENZOTHIAZOLES; BIOTRANSFORMATION; CARCINOGENS; LIVER; LIVER NEOPLASMS; MONOAMINE OXIDASE INHIBITORS; MUTAGENICITY TESTS; MUTAGENS; OXAZOLIDINONES; PRECANCEROUS CONDITIONS; RATS; SALMONELLA TYPHIMURIUM; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

BACTERIA (MICROORGANISMS); GYMNOMYZA SAMOENSIS; SALMONELLA; SALMONELLA TYPHIMURIUM; TYPHIMURIUM;

EID: 0034695110     PISSN: 13835718     EISSN: None     Source Type: Journal    
DOI: 10.1016/S1383-5718(00)00139-X     Document Type: Article

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