2-Substituted paullones: CDK1/cyclin B-inhibiting property and in vitro antiproliferative activity

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 6, 2000, Pages 567-569

  Kunick, Conrad ^a   Schultz, Christiane ^a   Lemcke, Thomas ^a   Zaharevitz, Daniel W ^b   Gussio, Rick ^b   Jalluri, Ravi K ^b   Sausville, Edward A ^b   Leost, Maryse ^c   Meijer, Laurent ^c  

^a UNIVERSITY OF HAMBURG   (Germany)

^b Developmental Therapeutics Program   (United States)

^c STATION BIOLOGIQUE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

9 TRIFLUOROMETHYLPAULLONE; BENZAZEPINE DERIVATIVE; CYCLIN B; CYCLIN DEPENDENT KINASE; ENZYME INHIBITOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTINEOPLASTIC ACTIVITY; ARTICLE; ASTERIAS; DRUG SYNTHESIS; ENZYME INHIBITION; GROWTH INHIBITION; HUMAN; HUMAN CELL; IN VITRO STUDY; NONHUMAN; OOCYTE; TUMOR CELL LINE;

ANIMALIA; ASTERIAS;

EID: 0034689596     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(00)00048-2     Document Type: Article

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