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Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 20, 2000, Pages 2283-2286

Tetrahydroisoquinoline derivatives containing a benzenesulfonamide moiety as potent, selective human β3 adrenergic receptor agonists

(12) Parmee, Emma R a Brockunier, Linda L a He, Jiafang a Singh, Suresh B a Candelore, Mari R a Cascieri, Margaret A a Deng, Liping a Liu, Yong a Tota, Laurie a Wyvratt, Matthew J a Fisher, Michael H a Weber, Ann E a

a MERCK RESEARCH LABORATORIES (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIOBESITY AGENT; BETA 3 ADRENERGIC RECEPTOR STIMULATING AGENT; BIPHENYL DERIVATIVE; TETRAHYDROISOQUINOLINE DERIVATIVE;

ARTICLE; DRUG EFFECT; DRUG POTENCY; DRUG RECEPTOR BINDING; METABOLIC RATE; OBESITY;

ADRENERGIC BETA-AGONISTS; AMIDES; DRUG DESIGN; HUMAN; ISOQUINOLINES; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PEPTIDES; RECEPTORS, ADRENERGIC, BETA-1; RECEPTORS, ADRENERGIC, BETA-2; RECEPTORS, ADRENERGIC, BETA-3; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0034675701 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(00)00459-5 Document Type: Article

Times cited : (21)

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