Anti-AIDS agents Part 41: Synthesis and anti-HIV activity of 3',4'-di-o-(-)-camphanoyl-(+)-cis-khellactone (DCK) lactam analogues

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 10, 2000, Pages 1003-1005

  Yang, Zheng Yu ^a   Xia, Yi ^a   Xia, Peng ^a   Brossi, Arnold ^a   Cosentino, L Mark ^b   Lee, Kuo Hsiung ^a  

^a University of North Carolina   (United States)

^b BBI Biotech Research Laboratories   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

KHELLACTONE; LACTAM DERIVATIVE; ZIDOVUDINE;

ACQUIRED IMMUNE DEFICIENCY SYNDROME; ARTICLE; CELL LINE; DRUG INHIBITION; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS; STRUCTURE ANALYSIS;

ANTI-HIV AGENTS; BICYCLO COMPOUNDS, HETEROCYCLIC; BIOCHEMISTRY; CAMPHOR; COUMARINS; DRUG EVALUATION, PRECLINICAL; HUMANS; LACTAMS; LYMPHOCYTES; QUINOLONES; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; RNA VIRUSES;

EID: 0034658588     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(00)00126-8     Document Type: Article

References (9)

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5. Yang, Z. Y.; Xia, Y.; Xia, P.; Cosentino, L. M.; Lee, K. H unpublished data.
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7. 10 635.2730, found 635.2733.
8. 1H NMR analysis of the bis-(-)-camphanic esters.
9. 4.