An intramolecular arylation route to the kinafluorenones

Tetrahedron Letters

Volumn 41, Issue 28, 2000, Pages 5317-5320

  Qabaja, Ghassan ^a   Jones, Graham B ^a  

^a NORTHEASTERN UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

KINAFLUORENONE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBIOTIC THERAPY; ANTIMICROBIAL THERAPY; ARTICLE; DRUG SYNTHESIS; MOLECULAR INTERACTION;

EID: 0034622328     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)00848-0     Document Type: Article

References (16)

1. CRC Handbook of Antibiotic Compounds; Berdy, J., Ed.; CRC Press: Boca Raton, 1980.
2. Koyama, H.; Kamikawa, T. Tetrahedron Lett.1997, 38, 3973; Gould, S. J.; Chen, J.; Cone, M. C.; Gore, M. P.; Melville, C. R.; Tamaya, N. J. Org. Chem. 1996, 61, 5720; Gould, S. J.; Melville, C. R.; Cone, M. C.; Chen, J.; Carney, J. R. J. Org. Chem. 1997, 62, 320.
3. Koyama, H.; Kamikawa, T. Tetrahedron Lett.1997, 38, 3973; Gould, S. J.; Chen, J.; Cone, M. C.; Gore, M. P.; Melville, C. R.; Tamaya, N. J. Org. Chem. 1996, 61, 5720; Gould, S. J.; Melville, C. R.; Cone, M. C.; Chen, J.; Carney, J. R. J. Org. Chem. 1997, 62, 320.
4. Koyama, H.; Kamikawa, T. Tetrahedron Lett.1997, 38, 3973; Gould, S. J.; Chen, J.; Cone, M. C.; Gore, M. P.; Melville, C. R.; Tamaya, N. J. Org. Chem. 1996, 61, 5720; Gould, S. J.; Melville, C. R.; Cone, M. C.; Chen, J.; Carney, J. R. J. Org. Chem. 1997, 62, 320.
5. Cone, M. C.; Hassan, A. M.; Gore, M. P.; Gould, S. J.; Borders, D. B.; Alluri, M. R. J. Org. Chem. 1994, 59, 1923; Gore, M. P.; Gould, S. J.; Weller, D. D. J. Org. Chem. 1992, 57, 2774.
6. Cone, M. C.; Hassan, A. M.; Gore, M. P.; Gould, S. J.; Borders, D. B.; Alluri, M. R. J. Org. Chem. 1994, 59, 1923; Gore, M. P.; Gould, S. J.; Weller, D. D. J. Org. Chem. 1992, 57, 2774.
7. Gore, M. P.; Gould, S. J.; Weller, D. D. J. Org. Chem. 1991, 56, 2289.
8. Gould, S. J.; Melville, C. R. Bioorg. Med. Chem. Lett. 1995, 5, 51.
9. For the phthalide annelation route, see: Hauser, F. M.; Zhou, M. J. Org. Chem. 1996, 61, 5722.
10. Ames, D. E.; Opalko, A. Synthesis 1983, 234.
11. Qabaja, G.; Perchellet, E.; Perchellet, J.; Jones, G. B. Tetrahedron Lett. 2000, 41, 3007-3010.
12. Mingos, D. M. P.; Baghurst, D. R. Chem. Soc. Rev. 1991, 20, 1.
13. For pioneering examples in organic synthesis, see: Giguere, R. J.; Bray, T. L.; Duncan, S. M.; Majetich, G. Tetrahedron Lett. 1986, 27, 4945.
14. For previous reports from this laboratory, see: Huber, R. S.; Jones, G. B. J. Org. Chem. 1992, 57, 5778; Jones, G. B.; Huber, R. S.; Chau, S. Tetrahedron 1993, 49, 369; Jones, G. B.; Chapman, B. J. J. Org. Chem. 1993, 58, 5558.
15. For previous reports from this laboratory, see: Huber, R. S.; Jones, G. B. J. Org. Chem. 1992, 57, 5778; Jones, G. B.; Huber, R. S.; Chau, S. Tetrahedron 1993, 49, 369; Jones, G. B.; Chapman, B. J. J. Org. Chem. 1993, 58, 5558.
16. For previous reports from this laboratory, see: Huber, R. S.; Jones, G. B. J. Org. Chem. 1992, 57, 5778; Jones, G. B.; Huber, R. S.; Chau, S. Tetrahedron 1993, 49, 369; Jones, G. B.; Chapman, B. J. J. Org. Chem. 1993, 58, 5558.