Probing the extended binding determinants of oligosaccharyl transferase with synthetic inhibitors of asparagine-linked glycosylation

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 3, 2000, Pages 281-284

  Ufret, Maria De L ^a   Imperiali, Barbara ^a  

^a MASSACHUSETTS INSTITUTE OF TECHNOLOGY   (United States)

Author keywords

Enzyme inhibitors; Glycopeptides glycoproteins; Glycosylation; Solid phase synthesis

Indexed keywords

ASPARAGINE; ASPARAGINE LINKED OLIGOSACCHARIDE; DRUG ANALOG; ENZYME INHIBITOR; GLYCOPEPTIDE; TRANSFERASE;

ARTICLE; BINDING AFFINITY; CHEMICAL MODIFICATION; DRUG SYNTHESIS; PROTEIN GLYCOSYLATION; PROTEIN INTERACTION; PROTEIN STRUCTURE;

AMINO ACID SEQUENCE; ASPARAGINE; GLYCOSYLATION; HEXOSYLTRANSFERASES; MEMBRANE PROTEINS; MOLECULAR PROBES; SUBSTRATE SPECIFICITY; TRANSFERASES;

EID: 0034615024     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00684-8     Document Type: Article

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