Synthesis and enzyme inhibitory activities of a series of lipidic diamine and aminoalcohol derivatives on cytosolic and secretory phospholipases A2

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 3, 2000, Pages 285-288

  Lucas, Rut ^a   Úbeda, Amalia ^a   Payá, Miguel ^a   Alves, Mario ^b   Olmo, Esther Del ^b   López, José L ^b   San Feliciano, Arturo ^b  

^a UNIVERSITY OF VALENCIA   (Spain)

^b UNIVERSITY OF SALAMANCA   (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

AMINOALCOHOL; APAMIN; BEE VENOM; DIAMINE DERIVATIVE; PANCREAS ENZYME; PHOSPHOLIPASE A2; RECOMBINANT ENZYME; SNAKE VENOM;

ARTICLE; BEE; CELL LINE; CYTOTOXICITY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; INHIBITION KINETICS; MACROPHAGE; MOUSE; NEUTROPHIL; NONHUMAN; SNAKE; STRUCTURE ACTIVITY RELATION; SWINE;

AMINO ALCOHOLS; ANIMALS; CELL LINE; CYTOSOL; DIAMINES; HUMANS; LIPIDS; MICE; PHOSPHOLIPASES A; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY;

APOIDEA; MURINAE; SERPENTES; SUS SCROFA;

EID: 0034614985     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00680-0     Document Type: Article

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