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Volumn 22, Issue 3, 2000, Pages 389-396

Effects of cholinesterase inhibitors on a two-component chained schedule performance in rats

Author keywords

Acetylcholinesterase inhibitors; Alzheimer's disease; Brightness discrimination; DRL DRH chained schedule; Heptylphysostigmine; Organophosphate poisoning; Physotigmine; Tacrine

Indexed keywords

CHOLINESTERASE INHIBITOR; HEPTYLPHYSOSTIGMINE; PHYSOSTIGMINE; TACRINE; UNCLASSIFIED DRUG;

EID: 0034612055     PISSN: 08920362     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0892-0362(99)00086-0     Document Type: Article
Times cited : (7)

References (50)
  • 1
    • 0011819520 scopus 로고
    • Enzyme inhibitors as substrates: Interaction of esterases with esters of organophosphorous and carbamic acids
    • A. Neuberger, & E.L. Tatum. Amsterdam: North Holland Publishing Company
    • Aldridge W.N., Reiner E. Enzyme inhibitors as substrates. Interaction of esterases with esters of organophosphorous and carbamic acids Neuberger A., Tatum E.L. Frontiers of Biology. 1972;123-146 North Holland Publishing Company, Amsterdam.
    • (1972) Frontiers of Biology , pp. 123-146
    • Aldridge, W.N.1    Reiner, E.2
  • 2
    • 0023899578 scopus 로고
    • Mechanisms of cholineresterase inhibition in senile dementia of the Alzheimer type: Clinical, pharmacological, and therapeutic aspects
    • Becker R., Giocobini E. Mechanisms of cholineresterase inhibition in senile dementia of the Alzheimer type. Clinical, pharmacological, and therapeutic aspects Drug Dev Rev. 12:1988;163-195.
    • (1988) Drug Dev Rev , vol.12 , pp. 163-195
    • Becker, R.1    Giocobini, E.2
  • 3
    • 0014759764 scopus 로고
    • The use of carbamates and atropine in the protection of animals against poisoning by 1,2,3-trimethylpropyl methylphosphonofluoridate
    • Berry W.K., Davis D.R. The use of carbamates and atropine in the protection of animals against poisoning by 1,2,3-trimethylpropyl methylphosphonofluoridate. Biochem Pharmacol. 19:1970;927-934.
    • (1970) Biochem Pharmacol , vol.19 , pp. 927-934
    • Berry, W.K.1    Davis, D.R.2
  • 6
    • 0029860968 scopus 로고    scopus 로고
    • Relationship between pharmacodynamic activity and cognitive effects of eptastigmine in patients with Alzheimer's disease
    • Canal N., Imbimbo B.P. Relationship between pharmacodynamic activity and cognitive effects of eptastigmine in patients with Alzheimer's disease. Clin Pharmacol Ther. 60:1996;218-228.
    • (1996) Clin Pharmacol Ther , vol.60 , pp. 218-228
    • Canal, N.1    Imbimbo, B.P.2
  • 7
    • 0028788545 scopus 로고
    • Effects of cholinesterases and clonidine coadministration on rat cortex neurotransmitters in vivo
    • Caudra G., Giacobini E. Effects of cholinesterases and clonidine coadministration on rat cortex neurotransmitters in vivo. J Pharmacol Exp Ther. 275:1995;228-236.
    • (1995) J Pharmacol Exp Ther , vol.275 , pp. 228-236
    • Caudra, G.1    Giacobini, E.2
  • 8
    • 0028341720 scopus 로고
    • Cholinesterase inhibitor effects on neurotransmitters in rat cortex in vivo
    • Caudra G., Summers K., Giacobini E. Cholinesterase inhibitor effects on neurotransmitters in rat cortex in vivo. J Pharmacol Exp Ther. 270:1984;277-284.
    • (1984) J Pharmacol Exp Ther , vol.270 , pp. 277-284
    • Caudra, G.1    Summers, K.2    Giacobini, E.3
  • 9
    • 0025131198 scopus 로고
    • Reversibility of the inhibition of acetylcholinerterase by tacrine
    • Dawson R.M. Reversibility of the inhibition of acetylcholinerterase by tacrine. Neurosci Lett. 118:1990;85-87.
    • (1990) Neurosci Lett , vol.118 , pp. 85-87
    • Dawson, R.M.1
  • 10
    • 0026005792 scopus 로고
    • The behavioral effects of heptylphysostigmine, a new cholinesterase inhibitor, in tests of long-term and working memory in rodents
    • Dawson G.R., Bentley G., Draper F., Rycroft W., Iversen S.D., Pagella P.G. The behavioral effects of heptylphysostigmine, a new cholinesterase inhibitor, in tests of long-term and working memory in rodents. Pharmacol Biochem Behav. 39:1991;856-871.
    • (1991) Pharmacol Biochem Behav , vol.39 , pp. 856-871
    • Dawson, G.R.1    Bentley, G.2    Draper, F.3    Rycroft, W.4    Iversen, S.D.5    Pagella, P.G.6
  • 12
    • 0024329466 scopus 로고
    • The effect of heptylphysostigmine, a new cholinesterase inhibitor, on the central cholinergic system of the rat
    • De Sarno P., Pomponi M., Giacobini E., Tang X.C., Williams E. The effect of heptylphysostigmine, a new cholinesterase inhibitor, on the central cholinergic system of the rat. Neurochem Res. 14:1989;971-977.
    • (1989) Neurochem Res , vol.14 , pp. 971-977
    • De Sarno, P.1    Pomponi, M.2    Giacobini, E.3    Tang, X.C.4    Williams, E.5
  • 13
    • 0023857396 scopus 로고
    • Further analysis of the neuropharmacological profile of 9-amino-1,2,3,4-tetrahydroacridine (THA), an alleged drug for the treatment of Alzheimer's disease
    • Drukarch B., Leysen J.E., Stoof J.C. Further analysis of the neuropharmacological profile of 9-amino-1,2,3,4-tetrahydroacridine (THA), an alleged drug for the treatment of Alzheimer's disease. Life Sci. 42:1988;1011-1017.
    • (1988) Life Sci , vol.42 , pp. 1011-1017
    • Drukarch, B.1    Leysen, J.E.2    Stoof, J.C.3
  • 15
    • 0027429837 scopus 로고
    • Brain selective inhibition of acetylcholinesterase: A novel approach to therapy for Alzheimer's disease
    • Enz A., Amstutz R., Boddeke H., Gmelin G., Malanowski J. Brain selective inhibition of acetylcholinesterase. A novel approach to therapy for Alzheimer's disease Prog Brain Res. 98:1993;431-438.
    • (1993) Prog Brain Res , vol.98 , pp. 431-438
    • Enz, A.1    Amstutz, R.2    Boddeke, H.3    Gmelin, G.4    Malanowski, J.5
  • 16
    • 0025907011 scopus 로고
    • Tacrine: A pharmacological review
    • Freeman S.E., Dawson R.M. Tacrine. A pharmacological review Prog Neurobiol. 36:1991;257-277.
    • (1991) Prog Neurobiol , vol.36 , pp. 257-277
    • Freeman, S.E.1    Dawson, R.M.2
  • 17
    • 0025821567 scopus 로고
    • Effectiveness of 1,2,3,4-tetrahydro-9-aminoacridine (THA) as a pretreatment drug for protection of mice from acute diisopropylfluorophosphate (DFP) intoxication
    • Galli A., Mori F. Effectiveness of 1,2,3,4-tetrahydro-9-aminoacridine (THA) as a pretreatment drug for protection of mice from acute diisopropylfluorophosphate (DFP) intoxication. Arch Toxicol. 65:1991;330-334.
    • (1991) Arch Toxicol , vol.65 , pp. 330-334
    • Galli, A.1    Mori, F.2
  • 18
    • 0024328888 scopus 로고
    • Hemicholinium-3 impairs spatial learning and the deficit is reversed by cholinomimetics
    • Hagan J.J., Jansen J.H.M., Brockkamp C.L.E. Hemicholinium-3 impairs spatial learning and the deficit is reversed by cholinomimetics. Psychopharmacol. 98:1989;347-356.
    • (1989) Psychopharmacol , vol.98 , pp. 347-356
    • Hagan, J.J.1    Jansen, J.H.M.2    Brockkamp, C.L.E.3
  • 19
    • 0021646861 scopus 로고
    • Toxicity of anticholinesterases: Interactions of pyridostigmine and physostigmine with soman
    • Harris L.W., Lennox W.J., Talbot B.G., Anderson D.R., Swanson D.R. Toxicity of anticholinesterases. Interactions of pyridostigmine and physostigmine with soman Drug Chem Toxicol. 7:1984;507-526.
    • (1984) Drug Chem Toxicol , vol.7 , pp. 507-526
    • Harris, L.W.1    Lennox, W.J.2    Talbot, B.G.3    Anderson, D.R.4    Swanson, D.R.5
  • 21
    • 0025370706 scopus 로고
    • Low dose tetrahydroaminoacridine (THA) improves cognitive function but does not affect brain acetylcholine in rats
    • Hodges J., Riberio A.M., Gary J.A., Marchbanks R.M. Low dose tetrahydroaminoacridine (THA) improves cognitive function but does not affect brain acetylcholine in rats. Pharmacol Biochem Behav. 36:1990;291-298.
    • (1990) Pharmacol Biochem Behav , vol.36 , pp. 291-298
    • Hodges, J.1    Riberio, A.M.2    Gary, J.A.3    Marchbanks, R.M.4
  • 23
    • 0026774392 scopus 로고
    • The long-lasting cholinesterase heptylphysostigmine attenuates the scopolamine-induced learning impairment of rats in a 14-unit T-maze
    • Iijima S., Greig M.H., Garofaol P., Spangler E.L., Heller B., Brossi A., Ingram D.K. The long-lasting cholinesterase heptylphysostigmine attenuates the scopolamine-induced learning impairment of rats in a 14-unit T-maze. Neurosci Lett. 144:1992;79-82.
    • (1992) Neurosci Lett , vol.144 , pp. 79-82
    • Iijima, S.1    Greig, M.H.2    Garofaol, P.3    Spangler, E.L.4    Heller, B.5    Brossi, A.6    Ingram, D.K.7
  • 24
    • 0027942542 scopus 로고
    • Effects of the centrally acting cholinesterase inhibitors tetrahydroaminoacridine and E2020 on the basal concentration of extracellular acetylcholine in the hippocampus of freely moving rats
    • Kawashima K., Sato A., Yoshizawa M., Fuji T., Fujimoto K., Suzuki T. Effects of the centrally acting cholinesterase inhibitors tetrahydroaminoacridine and E2020 on the basal concentration of extracellular acetylcholine in the hippocampus of freely moving rats. Naunyn-Schmied Arch Pharmacol. 350:1994;523-528.
    • (1994) Naunyn-Schmied Arch Pharmacol , vol.350 , pp. 523-528
    • Kawashima, K.1    Sato, A.2    Yoshizawa, M.3    Fuji, T.4    Fujimoto, K.5    Suzuki, T.6
  • 25
    • 0024465639 scopus 로고
    • Clinical pharmacology of tetrahydroaminoacridine: A possible therapeutic agent for Alzheimer's disease
    • Kumar V., Becker R.E. Clinical pharmacology of tetrahydroaminoacridine. A possible therapeutic agent for Alzheimer's disease Int J Clin Pharmacol Ther Toxicol. 10:1989;478-485.
    • (1989) Int J Clin Pharmacol Ther Toxicol , vol.10 , pp. 478-485
    • Kumar, V.1    Becker, R.E.2
  • 26
    • 0001307702 scopus 로고
    • The role of cholinesterase inhibitors in Alzheimer's disease
    • Lamy P.P. The role of cholinesterase inhibitors in Alzheimer's disease. CNS Drug. 1:1994;146-165.
    • (1994) CNS Drug , vol.1 , pp. 146-165
    • Lamy, P.P.1
  • 28
    • 0022198106 scopus 로고
    • Relationship between reversible acetylcholinestrerase inhibition and efficacy against soman lethality
    • Lennox W.J., Harris L.W., Talbot B.G., Anderson D.R. Relationship between reversible acetylcholinestrerase inhibition and efficacy against soman lethality. Life Sci. 37:1985;793-798.
    • (1985) Life Sci , vol.37 , pp. 793-798
    • Lennox, W.J.1    Harris, L.W.2    Talbot, B.G.3    Anderson, D.R.4
  • 29
    • 84951384024 scopus 로고
    • A simplified method of evaluating dose-effect experiments
    • Litchfield J.T., Wilcoxon E. A simplified method of evaluating dose-effect experiments. J Pharmacol Exp Ther. 96:1949;99-113.
    • (1949) J Pharmacol Exp Ther , vol.96 , pp. 99-113
    • Litchfield, J.T.1    Wilcoxon, E.2
  • 30
    • 0026354437 scopus 로고
    • Cholinolytic antagonism to the disruptive effects of oral low doses of pyridostigmine on simple discrimination performance in rats
    • Liu W.F. Cholinolytic antagonism to the disruptive effects of oral low doses of pyridostigmine on simple discrimination performance in rats. Pharmacol Biochem Behav. 40:1991;745-749.
    • (1991) Pharmacol Biochem Behav , vol.40 , pp. 745-749
    • Liu, W.F.1
  • 31
    • 0026592471 scopus 로고
    • Acute effects of oral low doses of pyridostigmine on simple visual discrimination and unconditioned consummatory acts in rats
    • Liu W.F. Acute effects of oral low doses of pyridostigmine on simple visual discrimination and unconditioned consummatory acts in rats. Pharmacol Biochem Behav. 41:1992;251-254.
    • (1992) Pharmacol Biochem Behav , vol.41 , pp. 251-254
    • Liu, W.F.1
  • 32
    • 0029980124 scopus 로고    scopus 로고
    • Effects of antimuscarinic antiparkinsonian drugs on brightness discrimination performance in rats
    • Liu W.F. Effects of antimuscarinic antiparkinsonian drugs on brightness discrimination performance in rats. Pharmacol Biochem Behav. 54:1996;425-430.
    • (1996) Pharmacol Biochem Behav , vol.54 , pp. 425-430
    • Liu, W.F.1
  • 33
    • 0013652365 scopus 로고
    • Behavioral effects of physotigmine as prophylaxis against organophosphate poisoning
    • Oct. 15, Taiwan, R. O. C., (in Chinese with English abstract).
    • W.F. Liu, J.H. Shih, Behavioral effects of physotigmine as prophylaxis against organophosphate poisoning, Proceedings of the Third National Conference on Science and Technology of National Defense, Oct. 15, 1994, Taiwan, R. O. C., pp. 263-271 (in Chinese with English abstract).
    • (1994) Proceedings of the Third National Conference on Science and Technology of National Defense , pp. 263-271
    • Liu, W.F.1    Shih, J.H.2
  • 34
    • 0026091609 scopus 로고
    • Differential effects of physostigmine and pilocarpine on the spatial memory deficits produced by two septo-hippocampal deafferentations
    • Matsuoka N., Maeda N., Ohkubo Y., Yamaguchi I. Differential effects of physostigmine and pilocarpine on the spatial memory deficits produced by two septo-hippocampal deafferentations. Brain Res. 559:1991;233-240.
    • (1991) Brain Res , vol.559 , pp. 233-240
    • Matsuoka, N.1    Maeda, N.2    Ohkubo, Y.3    Yamaguchi, I.4
  • 35
    • 0002555053 scopus 로고
    • Effect of carboxylesterase inhibition on carbamate protection against soman toxicity
    • D.M. Maxwell, K.M. Brech, D.D.E. Lenz, Effect of carboxylesterase inhibition on carbamate protection against soman toxicity, Proc Sixth Med Chem Def Biosci Rev (1987) 17-24.
    • (1987) Proc Sixth Med Chem Def Biosci Rev , pp. 17-24
    • Maxwell, D.M.1    Brech, K.M.2    Lenz, D.D.E.3
  • 36
    • 0027502112 scopus 로고
    • Cholinesterase inhibitor effects on extracellular acethylcholine in rat striatum
    • Messamore E., Organe N., Giacobini E. Cholinesterase inhibitor effects on extracellular acethylcholine in rat striatum. Neuropharmacol. 32:1993;291-296.
    • (1993) Neuropharmacol , vol.32 , pp. 291-296
    • Messamore, E.1    Organe, N.2    Giacobini, E.3
  • 37
    • 0027239591 scopus 로고
    • Cholinesterase inhibitor effects on extracellular acetylcholine in rat cortex
    • Messamore E., Warpman U., Ogane N., Giacobini E. Cholinesterase inhibitor effects on extracellular acetylcholine in rat cortex. Neuropharmacol. 8:1993;745-750.
    • (1993) Neuropharmacol , vol.8 , pp. 745-750
    • Messamore, E.1    Warpman, U.2    Ogane, N.3    Giacobini, E.4
  • 38
  • 39
    • 0024818025 scopus 로고
    • Correlation of brain levels of 9-amino-1,2,3,4-tetrahydroacridine (THA) with neurochemical and behavioral changes
    • Nielsen J.A., Mena E.E., Williams I.H., Nocerini M.R., Liston D. Correlation of brain levels of 9-amino-1,2,3,4-tetrahydroacridine (THA) with neurochemical and behavioral changes. Eur J Pharmacol. 173:1989;53-64.
    • (1989) Eur J Pharmacol , vol.173 , pp. 53-64
    • Nielsen, J.A.1    Mena, E.E.2    Williams, I.H.3    Nocerini, M.R.4    Liston, D.5
  • 40
    • 0024992639 scopus 로고
    • Present state and future development of the therapy of Alzheimer's disease
    • Pomponi M., Giacobini E., Brufani M. Present state and future development of the therapy of Alzheimer's disease. Aging. 2:1990;125-153.
    • (1990) Aging , vol.2 , pp. 125-153
    • Pomponi, M.1    Giacobini, E.2    Brufani, M.3
  • 41
    • 0027476710 scopus 로고
    • Effects of age and strain on working memory in mice as measured by win-shift paradigm
    • Reitzmann R.F., Kling A., Melchior C.L., Glasky A.J. Effects of age and strain on working memory in mice as measured by win-shift paradigm. Pharmacol Biochem Behav. 44:1993;805-807.
    • (1993) Pharmacol Biochem Behav , vol.44 , pp. 805-807
    • Reitzmann, R.F.1    Kling, A.2    Melchior, C.L.3    Glasky, A.J.4
  • 42
    • 0025300554 scopus 로고
    • The effects of THA on medial septal lesion-iduced memory defects
    • Kr P., Riekkinen J., Sirvio P., Riekkinen The effects of THA on medial septal lesion-iduced memory defects. Pharmacol Biochem Behav. 36:1990;237-241.
    • (1990) Pharmacol Biochem Behav , vol.36 , pp. 237-241
    • Kr, P.1    Riekkinen, J.2    Sirvio, P.3    Riekkinen4
  • 43
    • 0026512632 scopus 로고
    • Reversal of cognitive impairment by heptyl physostigmine, a long-lasting cholinesterase inhibitor, in primates
    • Rupniak N.M.J., Tye S.J., Brazell C., Heald A., Iversen S.D., Pagella P.G. Reversal of cognitive impairment by heptyl physostigmine, a long-lasting cholinesterase inhibitor, in primates. J Neurol Sci. 107:1992;246-249.
    • (1992) J Neurol Sci , vol.107 , pp. 246-249
    • Rupniak, N.M.J.1    Tye, S.J.2    Brazell, C.3    Heald, A.4    Iversen, S.D.5    Pagella, P.G.6
  • 44
    • 33746140058 scopus 로고
    • Clinical pharmacology of aminoacridines in Alzheimer's disease
    • Schneider L.S. Clinical pharmacology of aminoacridines in Alzheimer's disease. Neurol. 43:1993;S64-S79.
    • (1993) Neurol , vol.43
    • Schneider, L.S.1
  • 45
    • 0024347568 scopus 로고
    • In vivo dose response response relationship between physostigmine and cholineraerase activity in RBC and tissues of rats
    • Somani S.M., Dube S.N. In vivo dose response response relationship between physostigmine and cholineraerase activity in RBC and tissues of rats. Life Sci. 44:1989;1907-1915.
    • (1989) Life Sci , vol.44 , pp. 1907-1915
    • Somani, S.M.1    Dube, S.N.2
  • 47
    • 0027468207 scopus 로고
    • Differential effects of physostigmine and 1,2,3,4-tetrahydroacridine on the β-adrenoceptor transduction system
    • Vivas N.M., Badia A., Marmol F., Dierssen M. Differential effects of physostigmine and 1,2,3,4-tetrahydroacridine on the β-adrenoceptor transduction system. Eur J Pharmacol Mol Pharmacol Sec. 245:1993;9-13.
    • (1993) Eur J Pharmacol Mol Pharmacol Sec , vol.245 , pp. 9-13
    • Vivas, N.M.1    Badia, A.2    Marmol, F.3    Dierssen, M.4
  • 48
    • 0028316959 scopus 로고
    • Hepatotoxic effects of tacrine administration in patients with Alzheimer's disease
    • Watkins P.B., Zimmerman H.J., Knapp M.J., Gracon S.I., Lewis K.W. Hepatotoxic effects of tacrine administration in patients with Alzheimer's disease. J Amer Med Assoc. 271:1994;992-998.
    • (1994) J Amer Med Assoc , vol.271 , pp. 992-998
    • Watkins, P.B.1    Zimmerman, H.J.2    Knapp, M.J.3    Gracon, S.I.4    Lewis, K.W.5
  • 49
    • 0029613811 scopus 로고
    • The pharmacology of Alzheimer's disease based on the cholinergic hypothesis: An update
    • Weinstock M. The pharmacology of Alzheimer's disease based on the cholinergic hypothesis. An update Neurodegeneration. 4:1995;349-356.
    • (1995) Neurodegeneration , vol.4 , pp. 349-356
    • Weinstock, M.1
  • 50
    • 0028899957 scopus 로고
    • The behavioral effects of heptylphysostigmine on rats lesioned in the nucleus basalis
    • Waite J.J., Thal L.J. The behavioral effects of heptylphysostigmine on rats lesioned in the nucleus basalis. Neurosci Res. 21:1995;251-259.
    • (1995) Neurosci Res , vol.21 , pp. 251-259
    • Waite, J.J.1    Thal, L.J.2


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