Allosteric modulation of the rat adenosine A1 receptor: Differential effects on agonist and antagonist binding

Drug Development Research

Volumn 51, Issue 4, 2000, Pages 207-215

  Kourounakis, Angeliki P ^a   Visser, Corine ^b   De Groote, Miriam ^b   Ijzerman, Ad P ^b  

^a ARISTOTLE UNIVERSITY OF THESSALONIKI   (Greece)

^b LEIDEN UNIVERSITY   (Netherlands)

Author keywords

Agonist affinity; G protein coupled receptor; GTP; NaCl; NEM; PD81,723

Indexed keywords

2 AMINO 4,5 DIMETHYL 3 (3 TRIFLUOROMETHYLBENZOYL)THIOPHENE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; 8 CYCLOPENTYLTHEOPHYLLINE; ADENOSINE A1 RECEPTOR AGONIST; ADENOSINE A1 RECEPTOR ANTAGONIST; GUANOSINE TRIPHOSPHATE; N 0840; N ETHYLMALEIMIDE; N6 CYCLOPENTYL 9 METHYLADENINE; SODIUM CHLORIDE; SURAMIN; UNCLASSIFIED DRUG;

ALLOSTERISM; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG RECEPTOR BINDING; IC 50; MALE; NONHUMAN; RAT; RECEPTOR AFFINITY;

EID: 0034464124     PISSN: 02724391     EISSN: None     Source Type: Journal    
DOI: 10.1002/ddr.1     Document Type: Article

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