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Biochemistry

Volumn 39, Issue 30, 2000, Pages 8768-8781

Probing the S1/S1' substrate binding pocket geometry of HIV-1 protease with modified aspartic acid analogues

(6) Short III, G F a Laikhter, A L a Lodder, M a Shayo, Y a Arslan, T a Hecht, S M a

a UNIVERSITY OF VIRGINIA (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PROTEINASE; VIRUS ENZYME;

ARTICLE; BINDING SITE; CONTROLLED STUDY; ENZYME ACTIVE SITE; ENZYME SUBSTRATE COMPLEX; HUMAN IMMUNODEFICIENCY VIRUS 1; MOLECULAR INTERACTION; MOLECULAR RECOGNITION; NONHUMAN; PRIORITY JOURNAL;

ASPARTIC ACID; BINDING SITES; CATALYSIS; DIMERIZATION; EPOXY COMPOUNDS; HIV PROTEASE; HIV PROTEASE INHIBITORS; HUMANS; HYDROGEN-ION CONCENTRATION; KINETICS; MODELS, MOLECULAR; NITROPHENOLS; OLIGOPEPTIDES; PROTEIN CONFORMATION; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY; THERMODYNAMICS;

EID: 0034254518 PISSN: 00062960 EISSN: None Source Type: Journal
DOI: 10.1021/bi000214t Document Type: Article

Times cited : (28)

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