A practical approach to highly functionalized benzodihydrofurans

Tetrahedron Letters

Volumn 41, Issue 14, 2000, Pages 2269-2273

  Plotkin, Michael ^a   Chen, Sanyou ^a   Spoors, P Grant ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOFURAN DERIVATIVE; BROMINE DERIVATIVE; LITHIUM DERIVATIVE; N,N DIMETHYLFORMAMIDE;

ARTICLE; BROMINATION; CHEMICAL REACTION; CYCLIZATION; SYNTHESIS;

EID: 0034175576     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)00159-3     Document Type: Article

References (12)

1. (a) Elliot, J. D.; Lago, M. A.; Cousins, R. D.; Gao, A.; Leber, J. D.; Erhard, K. F.; Nambi, P.; Elshourbagy, N. A.; Kumar, C.; Lee, J. A.; Bean, J. W.; DeBrosse, C. W.; Eggleston, D. S.; Brooks, D. P.; Feuerstein, G.; Ruffolo Jr., R. R.; Weinstock, J.; Gleason, J. G.; Peishoff, C. E.; Ohlstein, E. H. J. Med. Chem. 1994, 37, 1553-1557.
2. (b) Endothelin Receptors: From the Gene to the Human; Ruffolo Jr., R. R., Ed.; CRC: Boca Raton, 1995.
3. Hammond, M. L.; Zambias, R. A.; Chang, M. N.; Jensen, N. P.; McDonald, J.; Thompson, K.; Boulton, D. A.; Kopka, I. E.; Hand, K. M.; Opas, E. E.; Luell, S.; Bach, T.; Davies, P.; MacIntyre, D. E.; Bonney, R. J.; Humes, J. L. J. Med. Chem. 1990, 33, 908-918.
4. (a) Paquette, L. A.; Schulze, M. M.; Bolin, D. G. J. Org. Chem. 1994, 59, 2043-2051.
5. (b) Alabaster, R. J.; Cottrel, I. F.; Hands, D.; Humphrey, G. R; Kennedy, D. J.; Wright H. B. Synthesis 1989, 8, 598-603.
6. Nichols, D. E.; Hoffman, A. J.; Oberlander, R. A.; Riggs, R. M.; J. Med. Chem. 1986, 29, 302-304; Monte, A. P.; Marona. D. L.; Parker, M. A.; Wainscott, D. B.; Nelson, D. L.; Nichols, D. E. J. Med. Chem. 1996, 39, 2953-2961.
7. Nichols, D. E.; Hoffman, A. J.; Oberlander, R. A.; Riggs, R. M.; J. Med. Chem. 1986, 29, 302-304; Monte, A. P.; Marona. D. L.; Parker, M. A.; Wainscott, D. B.; Nelson, D. L.; Nichols, D. E. J. Med. Chem. 1996, 39, 2953-2961.
8. Parham, W. E.; Jones, L. D.; Sayed, Y. A. J. Org. Chem. 1976, 41, 1184-1186.
9. Bradsher, C. K.; Reames, D. C. J. Org. Chem. 1981, 46, 1384-1388.
10. +.
11. +.
12. Unpublished results.