Tertiapin potently and selectively blocks muscarinic K+ channels in rabbit cardiac myocytes

Journal of Pharmacology and Experimental Therapeutics

Volumn 293, Issue 1, 2000, Pages 196-205

  Kitamura, Hidetsuna ^a,b   Yokoyama, Mitsuhiro ^b   Akita, Hozuka ^b   Matsushita, Kenji ^c   Kurachi, Yoshihisa ^c   Yamada, Mitsuhiko ^a  

^a NATIONAL CEREBRAL AND CARDIOVASCULAR CENTER   (Japan)

^b KOBE UNIVERSITY SCHOOL OF MEDICINE   (Japan)

^c OSAKA UNIVERSITY MEDICAL SCHOOL   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

CALCIUM CHANNEL; MUSCARINIC RECEPTOR; PEPTIDE DERIVATIVE; POTASSIUM CHANNEL; POTASSIUM CHANNEL BLOCKING AGENT; TERTIAPIN; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG INHIBITION; DRUG POTENCY; DRUG SELECTIVITY; HEART MUSCLE CELL; MALE; NONHUMAN; POTASSIUM CURRENT; PRIORITY JOURNAL; RABBIT;

AMINO ACID SEQUENCE; ANIMALS; ATP-BINDING CASSETTE TRANSPORTERS; BEE VENOMS; CELL MEMBRANE; CELL SEPARATION; ELECTROPHYSIOLOGY; G PROTEIN-COUPLED INWARDLY-RECTIFYING POTASSIUM CHANNELS; HEART; MALE; MEMBRANE POTENTIALS; MOLECULAR SEQUENCE DATA; MUSCARINIC ANTAGONISTS; MYOCARDIUM; PATCH-CLAMP TECHNIQUES; POTASSIUM CHANNEL BLOCKERS; POTASSIUM CHANNELS; POTASSIUM CHANNELS, INWARDLY RECTIFYING; RABBITS; RECEPTORS, MUSCARINIC;

EID: 0034115508     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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