Synthesis and antimalarial activities of base-catalyzed adducts of 11- azaartemisinin

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 5, 2000, Pages 1111-1116

  Mekonnen, Belew ^a   Weiss, Everett ^b   Katz, Esther ^b   Ma, Jingyuan ^b   Ziffer, Herman ^b   Kyle, Dennis E ^c  

^a NATIONAL INSTITUTE OF MENTAL HEALTH   (United States)

^b NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

^c WALTER REED ARMY INSTITUTE OF RESEARCH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETYLENE; ALKENE; ARTEMISININ; ARTEMISININ DERIVATIVE; BASE; NITRILE;

ANTIMALARIAL ACTIVITY; ARTICLE; CATALYSIS; CONJUGATION; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PLASMODIUM FALCIPARUM; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTIMALARIALS; AZA COMPOUNDS; CATALYSIS; MAGNETIC RESONANCE SPECTROSCOPY; PLASMODIUM FALCIPARUM; SESQUITERPENES;

PLASMODIUM FALCIPARUM;

EID: 0034086205     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00049-3     Document Type: Article

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