A new route to N-substituted 11-azaartemisinins

Tetrahedron Letters

Volumn 38, Issue 5, 1997, Pages 731-734

  Mekonnen, Belew ^a   Ziffer, Herman ^b  

^a NATIONAL INSTITUTE OF MENTAL HEALTH   (United States)

^b NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

11 AZAARTEMISININ DERIVATIVE; ANTIMALARIAL AGENT; ARTEMISININ DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; REACTION ANALYSIS;

EID: 0031016105     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(96)02417-3     Document Type: Article

References (7)

1. (a) Luo, X.-D. and Shen, C. C.; Med. Res. Rev. 1987, 7, 29.
2. (b) Jung, M.; Current Med. Chem. 1994, 1, 35.
3. Meshnick, S. R.; Thomas, A.; Ranz, A.; Xu, C.M. and H.-Z. Pan, H.-Z.; Mol. Biochem. Parasitol. 1991, 49, 181.
4. Torok, D. S. and Ziffer, H.; J. Med. Chem. 1995, 38, 5045.
5. Fang, F. G.; Prato, M.; Kim, G. and Danishefsky, S. J.; Tetrahedron Letters 1989, 30, 3625.
6. Dijkink, J.; Eriksen, K.; Goubitz, K.; van Zanden, M. N. A. and Hiemstra, H.; Tetrahedron Asymmetry 1996, 7, 515.
7. 3, 75.4 MHz) δ 13.2, 14.5, 20.1, 23.0, 25.4, 25.8, 33.0, 33.5, 34.0, 37.0, 37.9, 38.8, 45.9, 51.8, 60.8, 79.2, 80.5, 105.2, 172.2, 172.9.