(Partial) agonist/antagonist properties of novel diarylalkyl carbamates on histamine H3 receptors

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 5, 2000, Pages 1139-1149

  Sasse, Astrid ^a   Stark, Holger ^a   Ligneau, Xavier ^b   Elz, Sigurd ^a   Reidemeister, Sibylle ^a   Ganellin, C Robin ^c   Schwartz, Jean Charles ^d   Schunack, Walter ^a  

^a FREIE UNIVERSITÄT BERLIN   (Germany)

^b Laboratoire Bioprojet   (France)

^c UNIVERSITY COLLEGE LONDON   (United Kingdom)

^d INSERM   (France)

Author keywords

[No Author keywords available]

Indexed keywords

CARBAMIC ACID DERIVATIVE; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR AGONIST; HISTAMINE H3 RECEPTOR ANTAGONIST; LIGAND; PHOSGENE;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; BRAIN SYNAPTOSOME; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; HISTAMINE RELEASE; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

ANIMALS; CARBAMATES; HISTAMINE AGONISTS; HISTAMINE ANTAGONISTS; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; MICE; RATS; RECEPTORS, HISTAMINE H3;

ANIMALIA;

EID: 0034076460     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00050-X     Document Type: Article

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