Radiosynthesis of [14C]- and [3H]-robalzotan a selective 5-HT(1A) antagonist

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 43, Issue 5, 2000, Pages 437-447

  Werner, Tom F ^a   Sohn, Daniel ^a   Johansson, Rolf ^a  

^a ASTRAZENECA R AND D   (Sweden)

Author keywords

5HT(1A) antagonist; Palladium catalyzed carbonylation; Palladium catalyzed cyanylation; Robalzotan

Indexed keywords

CARBONYLATION; CARBOXYLATION; CATALYSIS; HYDROGENATION; PALLADIUM COMPOUNDS;

5HT(1A) ANTAGONIST; BENZOPYRANS; CARBON 14; CATALYTIC HYDROGENATION; PALLADIUM CATALYZED CARBONYLATION; PALLADIUM CATALYZED CYANYLATION; PALLADIUM-CATALYZED; RADIOSYNTHESIS; ROBALZOTAN; TRITIUM GAS;

TRITIUM;

BENZOPYRAN DERIVATIVE; CARBON 14; NITRILE; PALLADIUM; ROBALZOTAN; SEROTONIN 1A ANTAGONIST; TRITIUM;

ARTICLE; HYDROGENATION; HYDROLYSIS; ISOTOPE LABELING; SYNTHESIS;

TRITIUM;

EID: 0034071468     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(200004)43:5<437::AID-JLCR329>3.0.CO;2-J     Document Type: Article

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