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Volumn 115, Issue 5, 2000, Pages 271-279

Pharmacological and clinical aspects of fluvoxamine (Depromel®), the first selective serotonin reuptake inhibitor approved for clinical use employed in Japan

Author keywords

Depression; Depromel ; Fluvoxamine; Obsessive compulsive disorder (OCD); Selective serotonin reuptake inhibitor (SSRI)

Indexed keywords

ALPHA 1 ADRENERGIC RECEPTOR; FLUVOXAMINE; FLUVOXAMINE MALEATE; HISTAMINE H1 RECEPTOR; MUSCARINIC RECEPTOR; PLACEBO; SEROTONIN UPTAKE INHIBITOR; TRICYCLIC ANTIDEPRESSANT AGENT;

EID: 0034028180     PISSN: 00155691     EISSN: None     Source Type: Journal    
DOI: 10.1254/fpj.115.271     Document Type: Review
Times cited : (5)

References (50)
  • 1
    • 0017646651 scopus 로고
    • Fluvoxamine, a specific 5-hydroxytryptamine uptake inhibitor
    • Claassen V, Davies JE, Hertting G and Placheta P: Fluvoxamine, a specific 5-hydroxytryptamine uptake inhibitor. Br J Pharmacol 60, 505-516 (1977)
    • (1977) Br J Pharmacol , vol.60 , pp. 505-516
    • Claassen, V.1    Davies, J.E.2    Hertting, G.3    Placheta, P.4
  • 2
    • 0001875379 scopus 로고    scopus 로고
    • Drugs and the treatment of psychiatric disorders - Depression and mania
    • Edited by Hardman JG and Limbird LE, The McGraw-Hill Co, New York
    • th, ed. Edited by Hardman JG and Limbird LE, pp431-459, The McGraw-Hill Co, New York (1996)
    • (1996) th, Ed. , pp. 431-459
    • Baidessarini, R.J.1
  • 4
    • 85037957005 scopus 로고    scopus 로고
    • Japanese source
  • 5
    • 1542354940 scopus 로고
    • Masked depression in middle aged men
    • Krai VA: Masked depression in middle aged men. Can Med Assoc J 79, 1-5 (1958)
    • (1958) Can Med Assoc J , vol.79 , pp. 1-5
    • Krai, V.A.1
  • 6
    • 0000264756 scopus 로고
    • The catecholamine hypothesis of affective disorders; a review of supporting evidence
    • Schildkraut JJ: The catecholamine hypothesis of affective disorders; a review of supporting evidence. Am J Psychiatry 122, 509-522 (1965)
    • (1965) Am J Psychiatry , vol.122 , pp. 509-522
    • Schildkraut, J.J.1
  • 7
    • 0014150508 scopus 로고
    • The biochemistry of affective disorders
    • Coppen A: The biochemistry of affective disorders. Br J Psychiatry 113, 1237-1264 (1967)
    • (1967) Br J Psychiatry , vol.113 , pp. 1237-1264
    • Coppen, A.1
  • 8
    • 0000876391 scopus 로고
    • The treatment of depressive state with G 22355 (imipramine hydrochloride)
    • Kuhn R: The treatment of depressive state with G 22355 (imipramine hydrochloride). Am J Psychiatry 115, 459-464 (1958)
    • (1958) Am J Psychiatry , vol.115 , pp. 459-464
    • Kuhn, R.1
  • 9
    • 0014990917 scopus 로고
    • Endogenous depression with and without disturbances in the 5-hydroxy-tryptamine metabolism
    • Korf J and van Prag HM: Endogenous depression with and without disturbances in the 5-hydroxy-tryptamine metabolism. Psychopharmacologia 19, 148-152 (1971)
    • (1971) Psychopharmacologia , vol.19 , pp. 148-152
    • Korf, J.1    Van Prag, H.M.2
  • 10
    • 0022528874 scopus 로고
    • Consistent evidence for a biological subtype of depression characterized by low monoamine levels
    • Gibbons RD and Davis JM: Consistent evidence for a biological subtype of depression characterized by low monoamine levels. Acta Psychiatry Scand 74, 8-12 (1986)
    • (1986) Acta Psychiatry Scand , vol.74 , pp. 8-12
    • Gibbons, R.D.1    Davis, J.M.2
  • 12
    • 12944323386 scopus 로고    scopus 로고
    • Chapter 8, Drug treatments for obsessive compulsive disorder, panic disorder and phobic disorder
    • Cambridge University Press, Cambridge
    • Stahl SM: Chapter 8, Drug treatments for obsessive compulsive disorder, panic disorder and phobic disorder. In Essential Psychopharmacology "Neuroscientific Basis and Practical Applications" pp216-248, Cambridge University Press, Cambridge (1996)
    • (1996) Essential Psychopharmacology "Neuroscientific Basis and Practical Applications" , pp. 216-248
    • Stahl, S.M.1
  • 14
    • 0023501985 scopus 로고
    • Serotonergic responsivity in obsessive-compulsive disorder. Comparison of patients and health controls
    • Zohar J, Mueller EA, Insel TR, Zohar-Kadouch RC and Murphy DL: Serotonergic responsivity in obsessive-compulsive disorder. Comparison of patients and health controls. Arch Gen Psychiatry 44, 946-951 (1987)
    • (1987) Arch Gen Psychiatry , vol.44 , pp. 946-951
    • Zohar, J.1    Mueller, E.A.2    Insel, T.R.3    Zohar-Kadouch, R.C.4    Murphy, D.L.5
  • 16
    • 0028036323 scopus 로고
    • Regional cerebral blood flow measured during symptom provocation in obsessive-compulsive disorder using oxygen 15-labeled carbon dioxide and positron emission tomography
    • Rauch SL, Jenike MA, Alpert NM, Baer L, Breiter HCR, Savage CR and Fischman AJ: Regional cerebral blood flow measured during symptom provocation in obsessive-compulsive disorder using oxygen 15-labeled carbon dioxide and positron emission tomography. Arch Gen Psychiatry 51, 62-70 (1994)
    • (1994) Arch Gen Psychiatry , vol.51 , pp. 62-70
    • Rauch, S.L.1    Jenike, M.A.2    Alpert, N.M.3    Baer, L.4    Breiter, H.C.R.5    Savage, C.R.6    Fischman, A.J.7
  • 17
    • 0020536393 scopus 로고
    • Review of the animal pharmacology and pharmacokinetics of fluvoxamine
    • Claassen V: Review of the animal pharmacology and pharmacokinetics of fluvoxamine. Br J Clin Pharmacol 15, 349S-355S (1983)
    • (1983) Br J Clin Pharmacol , vol.15
    • Claassen, V.1
  • 18
    • 85037957726 scopus 로고    scopus 로고
    • Japanese source
  • 19
    • 85037952280 scopus 로고    scopus 로고
    • Japanese source
  • 20
    • 0032539862 scopus 로고    scopus 로고
    • Increase in the cerebrospinal fluid content of neurosteroids in patients with unipolar major depression who are receiving fluoxetine or fluvoxamine
    • Uzunova V, Sheline Y, Davis JM, Rasmussen A, Uzunov DP, Costa E and Guidotti A: Increase in the cerebrospinal fluid content of neurosteroids in patients with unipolar major depression who are receiving fluoxetine or fluvoxamine. Proc Natl Acad Sci USA 95, 3239-3244 (1998)
    • (1998) Proc Natl Acad Sci USA , vol.95 , pp. 3239-3244
    • Uzunova, V.1    Sheline, Y.2    Davis, J.M.3    Rasmussen, A.4    Uzunov, D.P.5    Costa, E.6    Guidotti, A.7
  • 21
    • 0028989563 scopus 로고
    • Neither the 5-HT1A- Nor 5-HT2-receptor subtype mediates the effect of fluvoxamine, a selective serotonin reuptake inhibitor, on forced-swimming-induced immobility in mice
    • Egawa T, Ichimaru Y, Imanishi T and Sawa A: Neither the 5-HT1A- nor 5-HT2-receptor subtype mediates the effect of fluvoxamine, a selective serotonin reuptake inhibitor, on forced-swimming-induced immobility in mice. Jpn J Pharmacol 68, 71-75 (1995)
    • (1995) Jpn J Pharmacol , vol.68 , pp. 71-75
    • Egawa, T.1    Ichimaru, Y.2    Imanishi, T.3    Sawa, A.4
  • 22
    • 85037968911 scopus 로고    scopus 로고
    • Japanese source
  • 23
    • 0025961370 scopus 로고
    • Evaluation of marbleburying behavior as a model of anxiety
    • Njung'e K and Handley SL: Evaluation of marbleburying behavior as a model of anxiety. Pharmacol Biochem Behav 38, 63-67 (1991)
    • (1991) Pharmacol Biochem Behav , vol.38 , pp. 63-67
    • Njung'e, K.1    Handley, S.L.2
  • 24
    • 0028989562 scopus 로고
    • 1A-receptor subtype mediates the effect of fluvoxamine, a selective serotonin reuptake inhibitor, on marbleburying behavior in mice
    • 1A-receptor subtype mediates the effect of fluvoxamine, a selective serotonin reuptake inhibitor, on marbleburying behavior in mice. Jpn J Pharmacol 68, 65-70 (1995)
    • (1995) Jpn J Pharmacol , vol.68 , pp. 65-70
    • Ichimaru, Y.1    Egawa, T.2    Sawa, A.3
  • 25
    • 8944249886 scopus 로고
    • In vitro pharmacology of fluvoxamine: Inhibition of monoamine uptake, receptor binding profile and functional receptor antagonism. Comparison with tricyclics and mianserin. Depression
    • Medidact
    • Tulp M, Mol F, Rademaker B and Schipper J: In vitro pharmacology of fluvoxamine: Inhibition of monoamine uptake, receptor binding profile and functional receptor antagonism. Comparison with tricyclics and mianserin. Depression, Anxiety and Aggression (Medidact), 9-19 (1988)
    • (1988) Anxiety and Aggression , pp. 9-19
    • Tulp, M.1    Mol, F.2    Rademaker, B.3    Schipper, J.4
  • 27
    • 85037956658 scopus 로고    scopus 로고
    • Japanese source
  • 28
    • 0029860967 scopus 로고    scopus 로고
    • Disposition of fluvoxamine in humans is determined by the polymorphic CYP2D6 and also by the CYP1A2 activity
    • Carrillo JA, Dahl MI, Svensson JO, Aim C, Rodriguez I and Bertilsson L: Disposition of fluvoxamine in humans is determined by the polymorphic CYP2D6 and also by the CYP1A2 activity. Clin Pharmacol Ther 60, 183-190 (1996)
    • (1996) Clin Pharmacol Ther , vol.60 , pp. 183-190
    • Carrillo, J.A.1    Dahl, M.I.2    Svensson, J.O.3    Aim, C.4    Rodriguez, I.5    Bertilsson, L.6
  • 30
    • 0031941954 scopus 로고    scopus 로고
    • Brain elimination half-life of fluvoxamine measured by 19F magnetic resonance spectroscopy
    • Strauss WL, Layton ME and Dager SR: Brain elimination half-life of fluvoxamine measured by 19F magnetic resonance spectroscopy. Am J Psychiatry 155, 380-384 (1998)
    • (1998) Am J Psychiatry , vol.155 , pp. 380-384
    • Strauss, W.L.1    Layton, M.E.2    Dager, S.R.3
  • 31
    • 0029976064 scopus 로고    scopus 로고
    • Newer antidepressants and the cytochrome P450 system
    • Nemeroff CB, DeVane CL and Pollock BG: Newer antidepressants and the cytochrome P450 system. Am J Psychiatry 153, 311-320 (1996)
    • (1996) Am J Psychiatry , vol.153 , pp. 311-320
    • Nemeroff, C.B.1    DeVane, C.L.2    Pollock, B.G.3
  • 33
    • 44049113266 scopus 로고
    • Influence of multiple-dose administration of fluvoxamine on the pharmacokinetics of the benzodiazepines bromazepam and lorazepam: A randomised, cross-over study
    • van Harten J, Holland RL and Wesnes K: Influence of multiple-dose administration of fluvoxamine on the pharmacokinetics of the benzodiazepines bromazepam and lorazepam: a randomised, cross-over study. Eur Neuropsychopharmacol 2, 381 (1992)
    • (1992) Eur Neuropsychopharmacol , vol.2 , pp. 381
    • Van Harten, J.1    Holland, R.L.2    Wesnes, K.3
  • 34
    • 0031901862 scopus 로고    scopus 로고
    • Safty of selegyline (deprenyl) in the treatment of Parkinson's disease
    • Heinonen EH and Myllyla V: Safty of selegyline (deprenyl) in the treatment of Parkinson's disease. Drug Saf 19, 11-22, (1998)
    • (1998) Drug Saf , vol.19 , pp. 11-22
    • Heinonen, E.H.1    Myllyla, V.2
  • 35
    • 0028333941 scopus 로고
    • Sertralinephenelzine drug interaction: A serotonin syndrome reaction
    • Graber MA, Hoehns TB and Perry PJ: Sertralinephenelzine drug interaction: a serotonin syndrome reaction. Ann Pharmacother 28, 732-735 (1994)
    • (1994) Ann Pharmacother , vol.28 , pp. 732-735
    • Graber, M.A.1    Hoehns, T.B.2    Perry, P.J.3
  • 36
    • 0027144398 scopus 로고
    • Serotonin syndrome induced fluvoxamine-lithium interaction
    • Ohman R and Spigset O: Serotonin syndrome induced fluvoxamine-lithium interaction. Pharmacopsychiatry 26, 263-264 (1993)
    • (1993) Pharmacopsychiatry , vol.26 , pp. 263-264
    • Ohman, R.1    Spigset, O.2
  • 37
    • 85037956420 scopus 로고    scopus 로고
    • Japanese source
  • 38
    • 85037970559 scopus 로고    scopus 로고
    • Japanese source
  • 39
    • 85037964534 scopus 로고    scopus 로고
    • Japanese source
  • 40
    • 85037960486 scopus 로고    scopus 로고
    • Japanese source
  • 41
    • 0031971040 scopus 로고    scopus 로고
    • Fluvoxamine prevents recurrence of depression: Results of a long-term, double-blind, placebo-controlled study
    • Terra JL and Montgomery SA: Fluvoxamine prevents recurrence of depression: results of a long-term, double-blind, placebo-controlled study. Int Clin Psychopharmacol 13, 55-62 (1998)
    • (1998) Int Clin Psychopharmacol , vol.13 , pp. 55-62
    • Terra, J.L.1    Montgomery, S.A.2
  • 42
    • 85037962605 scopus 로고    scopus 로고
    • Japanese source
  • 43
    • 85037958447 scopus 로고    scopus 로고
    • Japanese source
  • 44
    • 85037958973 scopus 로고    scopus 로고
    • Japanese source
  • 45
    • 0032126244 scopus 로고    scopus 로고
    • Effect of chronic antidepressant treatment on transcription factor binding activity in rat hippocampus and frontal cortex
    • Frechilla D, Otano A and Rio JD: Effect of chronic antidepressant treatment on transcription factor binding activity in rat hippocampus and frontal cortex. Prog Neuropsychopharmacol Biol Psychiatry 22, 787-802 (1998)
    • (1998) Prog Neuropsychopharmacol Biol Psychiatry , vol.22 , pp. 787-802
    • Frechilla, D.1    Otano, A.2    Rio, J.D.3
  • 46
    • 0022454164 scopus 로고
    • Effects of a selective 5-HT reuptake blocker, citalopram, on the sensitivity of 5-HT autoreceptors: Electrophysiological studies in the rat brain
    • Chaput Y, de Montigny C and Blier P: Effects of a selective 5-HT reuptake blocker, citalopram, on the sensitivity of 5-HT autoreceptors: electrophysiological studies in the rat brain. Naunyn Schmiedebergs Arch Pharmacol 333, 342-348 (1986)
    • (1986) Naunyn Schmiedebergs Arch Pharmacol , vol.333 , pp. 342-348
    • Chaput, Y.1    De Montigny, C.2    Blier, P.3
  • 47
    • 0028215631 scopus 로고
    • Effect of 21 days treatment with fluoxetine on stimulated endogenous 5-hydroxytryptamine overflow in the rat dosai raphe and sprachimastic nucleus studied using fast cyclic voltammetry in vitro
    • O'Connor JJ and Kruk ZL: Effect of 21 days treatment with fluoxetine on stimulated endogenous 5-hydroxytryptamine overflow in the rat dosai raphe and sprachimastic nucleus studied using fast cyclic voltammetry in vitro. Brain Res 640, 328-335 (1994)
    • (1994) Brain Res , vol.640 , pp. 328-335
    • O'Connor, J.J.1    Kruk, Z.L.2
  • 49
    • 0026750284 scopus 로고
    • Fluvoxamine in the treatment of demented elderly patients: A double-blined, placebo-controlled study
    • Olafsson K, Jorgensen S, Jensen HV, Bile A, Arup P and Andersen J: Fluvoxamine in the treatment of demented elderly patients: a double-blined, placebo-controlled study. Acta Psychiatr Scand 85, 453-456 (1992)
    • (1992) Acta Psychiatr Scand , vol.85 , pp. 453-456
    • Olafsson, K.1    Jorgensen, S.2    Jensen, H.V.3    Bile, A.4    Arup, P.5    Andersen, J.6
  • 50
    • 12944320517 scopus 로고    scopus 로고
    • Chapter 13 Other uses of the selective serotonin re-uptake inhibitors in psychiatry
    • Edited by Feighner JP and Boyer WF, John Wiley & Sons Ltd, New York
    • Boyer WF and Ewighner JP: Chapter 13 Other uses of the selective serotonin re-uptake inhibitors in psychiatry. In Advances in Basic Research and Clinical Practice, Second Edition, Edited by Feighner JP and Boyer WF, pp267-289, John Wiley & Sons Ltd, New York (1996)
    • (1996) Advances in Basic Research and Clinical Practice, Second Edition , pp. 267-289
    • Boyer, W.F.1    Ewighner, J.P.2


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