Prejunctional muscarinic inhibitory control of acetylcholine release in the human isolated detrusor: Involvement of the M4 receptor subtype

British Journal of Pharmacology

Volumn 129, Issue 3, 2000, Pages 493-500

  D'Agostino, Gianluigi ^a   Bolognesi, Maria L ^c   Lucchelli, Adele ^a   Vicini, Davide ^b   Balestra, Barbara ^c   Spelta, Valeria ^c   Melchiorre, Carlo ^c   Tonini, Marcello ^c  

^a UNIVERSITY OF PAVIA   (Italy)

^b General Hospital of Voghera   (Italy)

^c NONE

Author keywords

Human detrusor; Muscarinic receptor antagonists; Postjunctional muscarinic receptors; Prejunctional muscarinic autoreceptors; Smooth muscle contraction

Indexed keywords

4 DIPHENYLACETOXY 1 METHYLPIPERIDINE; 4 FLUOROHEXAHYDROSILADIPHENIDOL; ACETYLCHOLINE; ATROPINE; CHOLINE; HEXAMETHONIUM; MAMBA TOXIN 3; METHOCTRAMINE; MUSCARINIC M3 RECEPTOR; MUSCARINIC M4 RECEPTOR; MUSCARINIC RECEPTOR; MUSCARINIC RECEPTOR BLOCKING AGENT; MUSCARONE; PARAOXON; PHYSOSTIGMINE; PIRENZEPINE; RECEPTOR SUBTYPE; TETRODOTOXIN; TOXIN; TRIPINAMIDE; TRIPITRAMINE; UNCLASSIFIED DRUG;

ACETYLCHOLINE RELEASE; ADULT; AGED; ARTICLE; CHOLINERGIC NERVE; CONTROLLED STUDY; DETRUSOR MUSCLE; DRUG POTENCY; ELECTROSTIMULATION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN TISSUE; MALE; NEGATIVE FEEDBACK; NERVE ENDING; NEUROMUSCULAR SYNAPSE; PRIORITY JOURNAL; RECEPTOR AFFINITY; SMOOTH MUSCLE CONTRACTION;

EID: 0033972784     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0703080     Document Type: Article

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