Design, synthesis and binding at cloned muscarinic receptors of N-[5-(1'-substituted-acetoxymethyl)-3-oxadiazolyl] and N-[4-(1'-substituted-acetoxymethyl)-2-dioxolanyl] dialkyl amines

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 7, 2000, Pages 1559-1566

  Manfredini, Stefano ^a   Lampronti, Ilaria ^a   Vertuani, Silvia ^a   Solaroli, Nicola ^a   Recanatini, Maurizio ^b   Bryan, David ^c   Mckinney, Michael ^c  

^a UNIVERSITY OF FERRARA   (Italy)

^b UNIVERSITY OF BOLOGNA   (Italy)

^c MAYO CLINIC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1,3 DIOXOLANE DERIVATIVE; HEXAHYDROSILADIFENIDOL; MUSCARINIC M2 RECEPTOR; MUSCARINIC M3 RECEPTOR; MUSCARINIC M4 RECEPTOR; MUSCARINIC RECEPTOR; OXADIAZOLE DERIVATIVE;

ARTICLE; CATALYST; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG DESIGN; DRUG SYNTHESIS; HUNTINGTON CHOREA; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; PARKINSON DISEASE; STRUCTURE ACTIVITY RELATION;

AMINES; ANIMALS; CHO CELLS; CLONING, MOLECULAR; CRICETINAE; DIOXOLANES; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; MUSCARINIC ANTAGONISTS; OXADIAZOLES; RADIOLIGAND ASSAY; RECEPTORS, MUSCARINIC; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSFECTION;

EID: 0033936571     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00092-4     Document Type: Article

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