Piperazine analog of vesamicol: In vitro and in vivo characterization for vesicular acetylcholine transporter

Synapse

Volumn 38, Issue 1, 2000, Pages 27-37

  Bando, Kazunori ^a   Naganuma, Tomoyoshi ^a   Taguchi, Kazumi ^a   Ginoza, Yasushi ^a   Tanaka, Yoshitomo ^a   Koike, Katsuo ^b   Takatoku, Keizo ^a  

^a Daiichi Radioisotope Laboratories Ltd   (Japan)

^b TOHO UNIVERSITY   (Japan)

Author keywords

Autoradiography; Cholinergic; Radioiodinated ligand; Synaptic vesicle; Vesamicol

Indexed keywords

DRC 140; GUANIDINE DERIVATIVE; HALOPERIDOL; IODOBENZOVESAMICOL; PIPERAZINE DERIVATIVE; SIGMA OPIATE RECEPTOR; TRACER; TRANS 5 IODO 2 HYDROXY 3 [4 PHENYLPIPERAZINYL] TETRALIN; UNCLASSIFIED DRUG; VESAMICOL DERIVATIVE; VESICULAR ACETYLCHOLINE TRANSPORTER;

ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; BRAIN; CHOLINERGIC NERVE; CHOLINERGIC SYSTEM; CONTROLLED STUDY; CORPUS STRIATUM; DRUG BRAIN LEVEL; DRUG PROTEIN BINDING; DRUG SYNTHESIS; FRONTAL CORTEX; GUINEA PIG; HIPPOCAMPUS; ISOTOPE LABELING; MALE; NERVE FUNCTION; NONHUMAN; OCCIPITAL CORTEX; PRIORITY JOURNAL; RADIOACTIVITY; RAT; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY; SYNAPSE VESICLE;

ACETYLCHOLINE; ANIMALS; BRAIN; CARRIER PROTEINS; GUINEA PIGS; IODINE RADIOISOTOPES; MALE; MEMBRANE TRANSPORT PROTEINS; NEUROMUSCULAR DEPOLARIZING AGENTS; NEURONS; PIPERAZINES; PIPERIDINES; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; SUBCELLULAR FRACTIONS; SYNAPTIC VESICLES; TOMOGRAPHY, EMISSION-COMPUTED, SINGLE-PHOTON; VESICULAR ACETYLCHOLINE TRANSPORT PROTEINS; VESICULAR TRANSPORT PROTEINS;

EID: 0033845780     PISSN: 08874476     EISSN: None     Source Type: Journal    
DOI: 10.1002/1098-2396(200010)38:1<27::AID-SYN4>3.0.CO;2-1     Document Type: Article

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