Design and synthesis of acidic dipeptide hydroxamate inhibitors of procollagen C-proteinase

Journal of Peptide Science

Volumn 6, Issue 9, 2000, Pages 489-495

  Ovens, Annabel ^a,b   Joule, John A ^b   Kadler, Karl E ^a  

^a UNIVERSITY OF MANCHESTER   (United Kingdom)

^b UNIVERSITY OF MANCHESTER   (United Kingdom)

Author keywords

BMP 1; Collagen; Fibrosis; Matrix

Indexed keywords

ASPARTIC ACID; BB 3103; DIPEPTIDE DERIVATIVE; GLUTAMIC ACID; HYDROXAMIC ACID DERIVATIVE; MARIMASTAT; MATRIX METALLOPROTEINASE INHIBITOR; PROCOLLAGEN; PROCOLLAGEN C PROTEINASE; PROTEINASE INHIBITOR; UNCLASSIFIED DRUG;

ACIDITY; ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CARBOXY TERMINAL SEQUENCE; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME ACTIVE SITE; ENZYME ASSAY; ENZYME INHIBITION; HUMAN; HUMAN CELL; IC 50; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

AMINO ACID SEQUENCE; BONE MORPHOGENETIC PROTEINS; COLLAGEN; COMPARATIVE STUDY; CONSENSUS SEQUENCE; DIPEPTIDES; ELECTROPHORESIS, POLYACRYLAMIDE GEL; ENZYME INHIBITORS; HUMAN; HYDROXAMIC ACIDS; MATRIX METALLOPROTEINASES; METALLOENDOPEPTIDASES; MOLECULAR SEQUENCE DATA; MOLECULAR STRUCTURE; SUPPORT, NON-U.S. GOV'T;

ANIMALIA;

EID: 0033832622     PISSN: 10752617     EISSN: None     Source Type: Journal    
DOI: 10.1002/1099-1387(200009)6:9<489::AID-PSC282>3.0.CO;2-K     Document Type: Article

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