Human bradykinin B2 receptor is activated by kallikrein and other serine proteases

Molecular Pharmacology

Volumn 58, Issue 4, 2000, Pages 828-836

  Hecquet, Claudie ^a   Tan, Fulong ^a   Marcic, Branislav M ^a   Erdös, Ervin G ^a  

^a UNIVERSITY OF ILLINOIS   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ARACHIDONIC ACID; BRADYKININ; BRADYKININ B2 RECEPTOR; CALCIUM ION; CATHEPSIN G; ICATIBANT; SERINE PROTEINASE; TISSUE KALLIKREIN; TRITIUM; TRYPSIN;

ANIMAL CELL; ARACHIDONIC ACID METABOLISM; ARTICLE; CALCIUM MOBILIZATION; ENDOTHELIUM CELL; HUMAN; HUMAN CELL; HYPOTENSION; ISOTOPE LABELING; KALLIKREIN KININ SYSTEM; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION; SWINE;

EID: 0033803667     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.58.4.828     Document Type: Article

References (38)

1. Expression of rat kallikrein and epithelial polarity in transfected Madin-Darby canine kidney cells
2. Tissue specific expressions of kallikrein-related genes in the rat
3. Bioregulation of kinins: Kallikreins, kininogens, and kininases
4. Proteinase-activated receptors: New functions for old enzymes
5. Kallikrein-induced uterine contraction independent of kinin formation
6. Kallistatin is a potent new vasodilator
7. Binding of high molecular weight kininogen to human endothelial cells is mediated via a site within domains 2 and 3 of the urokinase receptor
8. Proteinase-activated receptors: Novel mechanisms of signaling by serine proteases
9. A micromethod for determination of bradykininogen under several condition
10. Receptors for bradykinin and kallidin
11. Potentiation of bradykinin actions by ACE inhibitors
12. Metabolism of bradykinin by peptidases in health and disease
13. Ein neues Kreislaufhormon und seine Wirkung
14. Antibodies to the α(q subfamily of guanine nucleotide-binding regulatory protein α subunits attenuate activation of phosphatidylinositol 4,5-bisphosphate hydrolysis by hormones
15. Kininogens
16. Cloning and pharmacological characterization of a human bradykinin (BK-2 receptor
17. Analysis of binding data
18. 'Mirror image' antagonists of thrombin-induced platelet activation based on thrombin receptor structure
19. The G proteins of the Gα(i and Gα(q family couple the bradykinin receptor to the release of endothelium-derived relaxing factor
20. Contribution of kinins to the cardiovascular actions of angiotensin-converting enzyme inhibitors
21. N-terminal amino acid sequence of human urinary kallikrein homology with other serine proteases
22. 2 receptor
23. Kallikreins and kinins - Some unanswered questions about system characteristics and roles in human disease
24. Potentiation of the actions of bradykinin by angiotensin I converting enzyme (ACE) inhibitors. The role of expressed human bradykinin B2 receptors and ACE in CHO cells
25. Proteolysis of the human platelet and endothelial cell thrombin receptor by neutrophil-derived cathepsin G
26. Endothelial cell thrombin receptors and PAR-2. Two protease-activated receptors located in a single cellular environment
27. Activation of human and rabbit prokallikrein by serine and metalloproteases
28. The physiological significance of bradykinin
29. Renal bradykinin receptors: Localization, transduction pathways and molecular basis for a possible pathological role
30. Site of kininogenase secretion in the dog nephron
31. Metabolism of substance P and bradykinin by human neutrophils
32. Purification of human prokallikrein. Identification of the site of activation by the metalloproteinase thermolysin
33. Effects of an angiotensin-converting-enzyme inhibitor, ramipril, on cardiovascular events in high-risk patients
34. Uber die Wirkung des Kallikreins auf den isolierten Darm und uber eine neue darmkontrahierende Substanz
35. Kallikrein and prekallikrein of the isolated basolateral membrane of rat kidney
36. Characterization of a dipeptide hydrolase (kinase II; angiotensin I converting enzyme)