Radiosynthesis of [18F]Lu29-024: A potential PET ligand for brain imaging of the serotonergic 5-HT2 receptor

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 10, 2000, Pages 2511-2518

  Sobrio, Franck ^a   Amokhtari, Mostafa ^a   Gourand, Fabienne ^a   Dhilly, Martine ^a   Dauphin, François ^b   Barré, Louisa ^a  

^a UNIVERSITÉ DE CAEN   (France)

^b GIP CYCERON   (France)

Author keywords

[No Author keywords available]

Indexed keywords

LU 29024; SEROTONIN 2 RECEPTOR; SEROTONIN 2A ANTAGONIST; UNCLASSIFIED DRUG; CARBON; DIAGNOSTIC AGENT; FLUORINATED HYDROCARBON; FLUORINE; INDOLE DERIVATIVE; LIGAND; LU29 024; LU29-024; PIPERIDINE DERIVATIVE; SEROTONIN RECEPTOR;

ARTICLE; BRAIN REGION; DRUG DISTRIBUTION; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOTOPE LABELING; LIGAND BINDING; POSITRON EMISSION TOMOGRAPHY; PURIFICATION; RADIOACTIVITY; RADIOISOTOPE DISTRIBUTION; REACTION ANALYSIS; ANIMAL; BRAIN; BRAIN LEVEL; CHEMISTRY; COMPUTER ASSISTED EMISSION TOMOGRAPHY; METABOLISM; RAT; SCINTISCANNING; SPRAGUE DAWLEY RAT; SYNTHESIS;

ANIMALS; BRAIN; BRAIN CHEMISTRY; CARBON ISOTOPES; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; FLUORINE RADIOISOTOPES; HYDROCARBONS, FLUORINATED; INDOLES; ISOTOPE LABELING; LIGANDS; PIPERIDINES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, SEROTONIN; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0033626577     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00181-4     Document Type: Article

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