Synthesis and anticonvulsant activity of 3-aryl-5H-2,3-benzodiazepine AMPA antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 14, 1999, Pages 1953-1956

  Anderson, Benjamin A ^a   Harn, Nancy K ^a   Hansen, Marvin M ^a   Harkness, Allen R ^a   Lodge, David ^a   Leander, J David ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMPA RECEPTOR ANTAGONIST; BENZODIAZEPINE DERIVATIVE;

ANIMAL EXPERIMENT; ANTICONVULSANT THERAPY; ARTICLE; DRUG EFFECT; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; MOUSE; NONHUMAN;

ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID; ANIMALS; ANTICONVULSANTS; BENZODIAZEPINES; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROSHOCK; MICE; SEIZURES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0033584177     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00315-7     Document Type: Article

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