Effects of tyrosine289phenylalanine mutation on binding and functional properties of the human tachykinin NK2 receptor stably expressed in Chinese hamster ovary cells

Biochemical Pharmacology

Volumn 57, Issue 8, 1999, Pages 899-906

  Renzetti, Anna Rita ^a   Catalioto, Rose Marie ^a   Carloni, Cristina ^a   Criscuoli, Marco ^a   Cucchi, Paola ^a   Giolitti, Alessandro ^a   Zappitelli, Sabrina ^a   Rotondaro, Luigi ^a   Maggi, Carlo Alberto ^a  

^a Menarini Ricerche ^*  (Italy)

Author keywords

Chinese hamster ovary cells; Guanosine 5' triphosphate; Inositol 1,4,5 trisphosphate; NK2 receptor; Phenoxybenzamine

Indexed keywords

GUANOSINE TRIPHOSPHATE; INOSITOL 1,4,5 TRISPHOSPHATE; NEPADUTANT; NEUROKININ 2 RECEPTOR; NEUROKININ A; NEUROKININ A [3-10][3 LYSINE 8 GLYCINE GAMMA LACTAM 9 LEUCINE]; NEUROKININ A [4-10][8 BETA ALANINE]; NEUROKININ B; NEUROKININ DERIVATIVE; PHENOXYBENZAMINE; SAREDUTANT; SUBSTANCE P; PHENYLALANINE; TACHYKININ; TYROSINE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; FEMALE; HUMAN; MUTANT; MUTATION; NONHUMAN; POINT MUTATION; PRIORITY JOURNAL; ANIMAL; BINDING COMPETITION; DRUG ANTAGONISM; GENETIC TRANSFECTION; GENETICS; HAMSTER; METABOLISM; PHYSIOLOGY; SIGNAL TRANSDUCTION;

ANIMALS; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; GUANOSINE TRIPHOSPHATE; HUMANS; INOSITOL 1,4,5-TRISPHOSPHATE; NEUROKININ A; PHENOXYBENZAMINE; PHENYLALANINE; POINT MUTATION; RECEPTORS, NEUROKININ-2; SIGNAL TRANSDUCTION; SUBSTANCE P; TACHYKININS; TRANSFECTION; TYROSINE;

EID: 0033560177     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(98)00373-6     Document Type: Article

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